Art

J-GLOBAL ID：200902212408314835   Reference number：07A0357854

On-Line Synthesis of Pseudopeptide Library Incorporating a Benzodiazepinone Turn Mimic: Biological Evaluation on MC1 Receptors

ベンゾジアゼピノンターン構造模倣単位を含む擬ペプチドライブラリのオンライン合成 MC1受容体に関する生物学的評価

Author (7)： VERDIE Pascal (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  SUBRA Gilles (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  FELIU Lidia (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  SANCHEZ Pierre (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  BERGE Gilbert (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  GARCIN Genevieve (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA) ,  MARTINEZ Jean (Lab. des Aminoacides, Peptides et Proteines (LAPP), Univ. Montpellier I et II, Montpellier, FRA)
Material： Journal of Combinatorial Chemistry  (J Comb Chem)
Volume： 9  Issue： 2  Page： 254-262  Publication year： Mar. 2007 
JST Material Number： W1756A  ISSN： 1520-4766  CODEN： JCCHFF  Document type： Article
Article type： 原著論文  Country of issue： United States (USA)  Language： ENGLISH (EN)

Thesaurus term： *peptide ,...
Semi thesaurus term： *antagonist ,...

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JST classification (3)： Seven-membered heterocyclic compounds  (CF07110I) ,  Production and application of antigens,antibodies,complements  (ED04030W) ,  Basic research of immunotherapeutic agents and blood preparations  (GW22010D)

Substance index (13)： (3S)-N-Methyl-3α-(acetylaminomethyl)-2,5(3H,4H)-dioxo-1H-1,4-benzodiazepine-4-acetamide ,  (3S)-N-Methyl-3α-[4-(acetylamino)butyl]-2,5(3H,4H)-dioxo-1H-1,4-benzodiazepine-4-acetamide ,  (Nle4)-α-MSH ,  N^α-Palmitoyl-His-D-Phe-Arg-Trp-NH₂ ,  N^α-[[(3S)-3α-(Palmitoylaminomethyl)-2,5(3H,4H)-dioxo-1H-1,4-benzodiazepine-4-yl]acetyl]-Arg-Trp-NH₂ ,  N-Acetyl-Nle-Ala-His-D-Phe-Arg-Trp-NH₂ ,  N-Acetyl-Nle-Ala-Arg-D-Phe-Arg-Trp-NH₂ ,  N^α-[[(3S)-3α-(N-Acetyl-Nle-Ala-Arg-aminomethyl)-2,5(3H,4H)-dioxo-8-chloro-1H-1,4-benzodiazepine-4-yl]acetyl]tryptophanamide ,  N-Acetyl-Nle-Ala-His-D-Phe-Arg-3-(2-naphthyl)-Ala-NH₂ ,  N^α-[[(3S)-3α-(N-Acetyl-Nle-Ala-aminomethyl)-2,5(3H,4H)-dioxo-1H-1,4-benzodiazepine-4-yl]acetyl]-Arg-3-(2-naphthyl)-Ala-NH₂ ,  N^α-[[(3S)-3α-(N-Acetyl-Nle-Ala-aminomethyl)-2,5(3H,4H)-dioxo-7-methyl-1H-1,4-benzodiazepine-4-yl]acetyl]-Arg-3-(2-naphthyl)-Ala-NH₂ ,  N^α-[[(3S)-3α-[4-(N-Acetyl-Nle-Ala-amino)butyl]-2,5(3H,4H)-dioxo-1H-1,4-benzodiazepine-4-yl]acetyl]-Arg-3-(2-naphthyl)-Ala-NH₂ ,  N^α-[[(3S)-3α-[4-(N-Acetyl-Nle-Ala-amino)butyl]-2,5(3H,4H)-dioxo-7-methyl-1H-1,4-benzodiazepine-4-yl]acetyl]-Arg-3-(2-naphthyl)-Ala-NH₂

Terms in the title (5)： 模倣 ,  ペプチドライブラリ ,  オンライン ,  受容体 ,  生物学的評価