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J-GLOBAL ID：201702290335815872   Reference number：17A0503858

Yb(OTf)₃-CATALYZED SYNTHESIS OF 2-SUBSTITUTED 4(3H)-QUINAZOLINONES VIA CLEAVAGE OF A CARBON-CARBON BOND

炭素-炭素結合の開裂による2置換4(3H)-キナゾリノンのYb(OTf)₃触媒合成

Author (7)： YOSHIMURA Tsutomu (Kyoto Univ., Kyoto, JPN) ,  NAITO Shun-ichi (Kyoto Univ., Kyoto, JPN) ,  YUANJUN Di (Kyoto Univ., Kyoto, JPN) ,  SON Aoi (Kyoto Univ., Kyoto, JPN) ,  KIMURA Yu (Kyoto Univ., Kyoto, JPN) ,  TOSHIMITSU Akio (Kyoto Univ., Kyoto, JPN) ,  KONDO Teruyuki (Kyoto Univ., Kyoto, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 93  Issue： 2  Page： 816-823  Publication year： Apr. 01, 2016 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 原著論文  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： *cyclization reaction ,  diketone ,  one-pot synthesis ,  C-C bond ,  catalytic reaction ,  *cleavage reaction ,  nitrogen heterocyclic compound ,  polynuclear aromatic compound ,  carboxamide ,  aromatic carboxylic acid ,  aromatic ketone ,  aromatic amine ,  aminocarboxylic acid ,  aliphatic ketone ,  aliphatic carboxylic acid ,  carboxylate(ester) ,  keto acid
Semi thesaurus term： quinazolines ,  Benzamides

JST classification (1)： Pyrimidines  (CF07103W)

Substance index (13)： Dibenzoylmethane ,  Benzoylacetone ,  2-Amino-4-methylbenzamide ,  2-Amino-5-chlorobenzamide ,  2-Amino-5-methoxybenzamide ,  2-Amino-6-fluorobenzamide ,  2-Aminobenzamide ,  2-Methylquinazolin-4(3H)-one ,  2-Methyl-5-fluoro-4(3H)-quinazolinone ,  2-Methyl-6-chloro-4(3H)-quinazolinone ,  2-Methyl-6-methoxy-4(3H)-quinazolinone ,  2-Methyl-7-methyl-4(3H)-quinazolinone ,  Acetoacetic acid methyl

Reference (13)：

• For a review, see: (a) A. Will and J. Bergman, Curr. Org. Chem., 2003, 7, 659; (b) S. B. Mhaske and N. P. Argade, Tetrahedron, 2006, 62, 9787; (c) M. Demeunynck and I. Baussanne, Curr. Med. Chem., 2013, 20, 794; (d) I. Khan, A. Ibrar, W. Ahmed, and A. Saeed, Eur. J. Med. Chem., 2015, 90, 124.
• For a review, see: (a) D. J. Connolly, D. Cusack, T. P. O'Sullivan, and P. J. Guiry, Tetrahedron, 2005, 61, 10153; (b) L. He, H. Li, J. Chen, and X.-F. Wu, RSC Adv., 2014, 4, 12065.
• S. Niementowski, Ber., 1894, 27, 1394.
• M. S. Manhas, S. G. Amin, and V. V. Rao, Synthesis, 1977, 309.
• O. A. Maloshitskaya, J. Sinkkonen, V. V. Alekseyev, K. N. Zelenin, and K. Pihlaja, Tetrahedron, 2005, 61, 7294.

Terms in the title (7)： 炭素-炭素結合 ,  開裂 ,  置換 ,  キナゾリノン ,  Yb ,  OTF ,  触媒合成