文献
J-GLOBAL ID:201002293148137200
整理番号:10A0615609
強力にスムーズ化されたアンタゴニストとしての1-ピペラジニル-4-アリールフタラジンの設計
Design of 1-piperazinyl-4-arylphthalazines as potent Smoothened antagonists
著者 (23件):
LUCAS Brian S.
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
AARON Wade
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
AN Songzhu
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
AUSTIN Richard J.
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
BROWN Matthew
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
CHAN Hon
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
CHONG Angela
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
HUNGATE Randall
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
HUANG Tom
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
JIANG Ben
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
JOHNSON Michael G.
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
KAIZERMAN Jacob A.
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
LEE Gary
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
MCMINN Dustin L.
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
ORF Jessica
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
POWERS Jay P.
(Dep. of Medicinal Chemistry, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
RONG Minqing
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
TOTEVA Maria M.
(Dep. of Small Molecule Process and Product Dev., AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
UYEDA Craig
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
WICKRAMASINGHE Dineli
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
XU Guifen
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
YE Qiuping
(Dep. of Pharmacokinetics and Drug Metabolism, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
,
ZHONG Wendy
(Dep. of Oncology, AMGEN, 1120 Veterans Blvd., S. San Francisco, CA 94080, USA)
資料名:
Bioorganic & Medicinal Chemistry Letters
(Bioorganic & Medicinal Chemistry Letters)
巻:
20
号:
12
ページ:
3618-3622
発行年:
2010年06月15日
JST資料番号:
W0248A
ISSN:
0960-894X
資料種別:
逐次刊行物 (A)
発行国:
オランダ (NLD)
言語:
英語 (EN)