文献
J-GLOBAL ID:201202237473097491
整理番号:12A1646516
チオフェンカルボキサミド尿素の構造ベースの設計と最適化による,チェックポイントキナーゼ阻害剤(S)-5-(3-フルオロフェニル)-N-(ピペリジン-3-イル)-3-ウレイドチオフェン-2-カルボキサミド(AZD7762)の発見
Discovery of Checkpoint Kinase Inhibitor (S)-5-(3-Fluorophenyl)-N-(piperidin-3-yl)-3-ureidothiophene-2-carboxamide (AZD7762) by Structure-Based Design and Optimization of Thiophenecarboxamide Ureas
著者 (25件):
OZA Vibha
(AstraZeneca R&D Boston, Massachusetts, USA)
,
ASHWELL Susan
(AstraZeneca R&D Boston, Massachusetts, USA)
,
ALMEIDA Lynsie
(AstraZeneca R&D Boston, Massachusetts, USA)
,
BRASSIL Patrick
(AstraZeneca R&D Boston, Massachusetts, USA)
,
BREED Jason
(AstraZeneca R&D Alderley, Cheshire, GBR)
,
DENG Chun
(AstraZeneca R&D Boston, Massachusetts, USA)
,
GERO Thomas
(AstraZeneca R&D Boston, Massachusetts, USA)
,
GRONDINE Michael
(AstraZeneca R&D Boston, Massachusetts, USA)
,
HORN Candice
(AstraZeneca R&D Boston, Massachusetts, USA)
,
IOANNIDIS Stephanos
(AstraZeneca R&D Boston, Massachusetts, USA)
,
LIU Dongfang
(AstraZeneca R&D Boston, Massachusetts, USA)
,
LYNE Paul
(AstraZeneca R&D Boston, Massachusetts, USA)
,
NEWCOMBE Nicholas
(AstraZeneca R&D Alderley, Cheshire, GBR)
,
PASS Martin
(AstraZeneca R&D Alderley, Cheshire, GBR)
,
READ Jon
(AstraZeneca R&D Alderley, Cheshire, GBR)
,
READY Shannon
(AstraZeneca R&D Boston, Massachusetts, USA)
,
ROWSELL Sian
(AstraZeneca R&D, Macclesfield, GBR)
,
SU Mei
(AstraZeneca R&D Boston, Massachusetts, USA)
,
TOADER Dorin
(AstraZeneca R&D Boston, Massachusetts, USA)
,
VASBINDER Melissa
(AstraZeneca R&D Boston, Massachusetts, USA)
,
YU Dingwei
(AstraZeneca R&D Boston, Massachusetts, USA)
,
YU Yan
(AstraZeneca R&D Boston, Massachusetts, USA)
,
XUE Yafeng
(AstraZeneca R&D Moelndal, Moelndal, SWE)
,
ZABLUDOFF Sonya
(AstraZeneca R&D Boston, Massachusetts, USA)
,
JANETKA James
(AstraZeneca R&D Boston, Massachusetts, USA)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
55
号:
11
ページ:
5130-5142
発行年:
2012年06月14日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)