文献
J-GLOBAL ID:201302240786190563
整理番号:13A0775524
強力かつ経口効果的なTGR5作動薬としての4-フェノキシニコチンアミドおよび4-フェノキシピリミジン-5-カルボキサミド誘導体の設計,合成および抗糖尿病活性
Design, Synthesis, and Antidiabetic Activity of 4-Phenoxynicotinamide and 4-Phenoxypyrimidine-5-carboxamide Derivatives as Potent and Orally Efficacious TGR5 Agonists
著者 (9件):
DUAN Hongliang
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
NING Mengmeng
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
CHEN Xiaoyan
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
ZOU Qingan
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
ZHANG Liming
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
FENG Ying
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
ZHANG Lina
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
LENG Ying
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
,
SHEN Jianhua
(State Key Lab. of Drug Res., Shanghai Inst. of Materia Medica (SIMM), Chinese Acad. of Sci., Shanghai, CHN)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
55
号:
23
ページ:
10475-10489
発行年:
2012年12月13日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)