文献
J-GLOBAL ID:201402264680805988
整理番号:14A0451006
サイクリン依存的キナーゼ4(CDK4)およびAMPK関連キナーゼ5(ARK5)の強力阻害剤としての8-シクロペンチル-2-[4-(4-メチル-ピペラジン-1-イル)-フェニルアミノ]-7-オキソ-7,8-ジヒドロ-ピリド[2,3-d]ピリミジン-6-カルボニトリル(7x)の発見
Discovery of 8-Cyclopentyl-2-[4-(4-methyl-piperazin-1-yl)-phenylamino]-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidine-6-carbonitrile (7x) as a Potent Inhibitor of Cyclin-Dependent Kinase 4 (CDK4) and AMPK-Related Kinase 5 (ARK5)
著者 (13件):
REDDY M.V.Ramana
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
AKULA Balireddy
(Onconova Therapeutics Inc., Pennsylvania, USA)
,
COSENZA Stephen C.
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
ATHULURIDIVAKAR Saikrishna
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
MALLIREDDIGARI Muralidhar R.
(Onconova Therapeutics Inc., Pennsylvania, USA)
,
PALLELA Venkat R.
(Onconova Therapeutics Inc., Pennsylvania, USA)
,
BILLA Vinay K.
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
SUBBAIAH D.R.C.Venkata
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
BHARATHI E.Vijaya
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
VASQUEZ-DEL CARPIO Rodrigo
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
PADGAONKAR Amol
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
BAKER Stacey J.
(Icahn School of Medicine at Mount Sinai, New York, USA)
,
REDDY E.Premkumar
(Icahn School of Medicine at Mount Sinai, New York, USA)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
57
号:
3
ページ:
578-599
発行年:
2014年02月13日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)