文献
J-GLOBAL ID:201502201610988003
整理番号:15A1328323
強力で経口的にバイオアベイラビリティ選択的エストロゲン受容体ダウンレギュレーターおよびアンタゴニストである(E)-3-(3,5-ジフルオロ-4-((1R,3R)-2-(2-フルオロ-2-メチルプロピル)-3-メチル-2,3,4,9-テトラヒドロ-1H-ピリド[3,4-b]インドール-1-イル)フェニル)アクリル酸(AZD9496)への新規結合性モチーフの最適化
Optimization of a Novel Binding Motif to (E)-3-(3,5-Difluoro-4-((1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)phenyl)acrylic Acid (AZD9496), a Potent and Orally Bioavailable Selective Estrogen Receptor Downregulator and Antagonist
著者 (28件):
DE SAVI Chris
(AstraZeneca, Macclesfield, GBR)
,
DE SAVI Chris
(AstraZeneca R&D Boston, Massachusetts, USA)
,
BRADBURY Robert H.
(AstraZeneca, Macclesfield, GBR)
,
RABOW Alfred A.
(AstraZeneca, Macclesfield, GBR)
,
NORMAN Richard A.
(AstraZeneca, Macclesfield, GBR)
,
DE ALMEIDA Camila
(AstraZeneca, Macclesfield, GBR)
,
ANDREWS David M.
(AstraZeneca, Macclesfield, GBR)
,
BALLARD Peter
(AstraZeneca, Macclesfield, GBR)
,
BUTTAR David
(AstraZeneca, Macclesfield, GBR)
,
CALLIS Rowena J.
(AstraZeneca, Macclesfield, GBR)
,
CURRIE Gordon S.
(AstraZeneca, Macclesfield, GBR)
,
CURWEN Jon O.
(AstraZeneca, Macclesfield, GBR)
,
DAVIES Chris D.
(AstraZeneca, Macclesfield, GBR)
,
DONALD Craig S.
(AstraZeneca, Macclesfield, GBR)
,
FERON Lyman J. L.
(AstraZeneca, Macclesfield, GBR)
,
GINGELL Helen
(AstraZeneca, Macclesfield, GBR)
,
GLOSSOP Steven C.
(AstraZeneca, Macclesfield, GBR)
,
HAYTER Barry R.
(AstraZeneca, Macclesfield, GBR)
,
HUSSAIN Syeed
(AstraZeneca, Macclesfield, GBR)
,
KAROUTCHI Galith
(AstraZeneca, Macclesfield, GBR)
,
LAMONT Scott G.
(AstraZeneca, Macclesfield, GBR)
,
MACFAUL Philip
(AstraZeneca, Macclesfield, GBR)
,
MOSS Thomas A.
(AstraZeneca, Macclesfield, GBR)
,
PEARSON Stuart E.
(AstraZeneca, Macclesfield, GBR)
,
TONGE Michael
(AstraZeneca, Macclesfield, GBR)
,
WALKER Graeme E.
(AstraZeneca, Macclesfield, GBR)
,
WEIR Hazel M.
(AstraZeneca, Macclesfield, GBR)
,
WILSON Zena
(AstraZeneca, Macclesfield, GBR)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
58
号:
20
ページ:
8128-8140
発行年:
2015年10月22日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)