文献
J-GLOBAL ID:201502220586526316
整理番号:15A1184687
2-[1-(4,4-ジフルオロシクロヘキシル)ピペリジン-4-イル]-6-フルオロ-3-オキソ-2,3-ジヒドロ-1H-イソインドール-4-カルボアミド(NMS-P118)の発見:癌治療に対して強力で経口利用できる高度に選択的なPARP-1阻害剤
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1H-isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy
著者 (29件):
PAPEO Gianluca
(Nerviano Medical Sci. Srl, Milan, ITA)
,
POSTERI Helena
(Nerviano Medical Sci. Srl, Milan, ITA)
,
BORGHI Daniela
(Nerviano Medical Sci. Srl, Milan, ITA)
,
BUSEL Alina A.
(Chemical Diversity Res. Inst., Moscow Region, RUS)
,
CAPRERA Francesco
(Nerviano Medical Sci. Srl, Milan, ITA)
,
CASALE Elena
(Nerviano Medical Sci. Srl, Milan, ITA)
,
CIOMEI Marina
(Nerviano Medical Sci. Srl, Milan, ITA)
,
CIRLA Alessandra
(Nerviano Medical Sci. Srl, Milan, ITA)
,
CORTI Emiliana
(Nerviano Medical Sci. Srl, Milan, ITA)
,
D’ANELLO Matteo
(Nerviano Medical Sci. Srl, Milan, ITA)
,
FASOLINI Marina
(Nerviano Medical Sci. Srl, Milan, ITA)
,
FORTE Barbara
(Nerviano Medical Sci. Srl, Milan, ITA)
,
GALVANI Arturo
(Nerviano Medical Sci. Srl, Milan, ITA)
,
ISACCHI Antonella
(Nerviano Medical Sci. Srl, Milan, ITA)
,
KHVAT Alexander
(Chemical Diversity Res. Inst., Moscow Region, RUS)
,
KRASAVIN Mikhail Y.
(Chemical Diversity Res. Inst., Moscow Region, RUS)
,
LUPI Rosita
(Nerviano Medical Sci. Srl, Milan, ITA)
,
ORSINI Paolo
(Nerviano Medical Sci. Srl, Milan, ITA)
,
PEREGO Rita
(Nerviano Medical Sci. Srl, Milan, ITA)
,
PESENTI Enrico
(Nerviano Medical Sci. Srl, Milan, ITA)
,
PEZZETTA Daniele
(Accelera Srl, Milan, ITA)
,
RAINOLDI Sonia
(Nerviano Medical Sci. Srl, Milan, ITA)
,
RICCARDI-SIRTORI Federico
(Nerviano Medical Sci. Srl, Milan, ITA)
,
SCOLARO Alessandra
(Nerviano Medical Sci. Srl, Milan, ITA)
,
SOLA Francesco
(Nerviano Medical Sci. Srl, Milan, ITA)
,
ZUCCOTTO Fabio
(Nerviano Medical Sci. Srl, Milan, ITA)
,
FELDER Eduard R.
(Nerviano Medical Sci. Srl, Milan, ITA)
,
DONATI Daniele
(Nerviano Medical Sci. Srl, Milan, ITA)
,
MONTAGNOLI Alessia
(Nerviano Medical Sci. Srl, Milan, ITA)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
58
号:
17
ページ:
6875-6898
発行年:
2015年09月10日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)