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J-GLOBAL ID:201702250709762193   整理番号:17A1485548

強力な抗酸化活性を示すPPARα/γ作動薬としてのクマリンカルコンフィブレート系薬剤の新規構造クラス:設計,合成,生物学的評価および分子ドッキング研究【Powered by NICT】

A novel structural class of coumarin-chalcone fibrates as PPARα/γ agonists with potent antioxidant activities: Design, synthesis, biological evaluation and molecular docking studies
著者 (11件):
Niu Handong
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Niu Handong
(Center for Drug Evaluation, China Food and Drug Administration, NO.1 of Fuxing Road, Haidian District, Beijing 100038, People’s Republic of China)
Wang Wenbao
(Department of Natural Products Chemistry, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Li Jinyan
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Lei Yu
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Zhao Yong
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Yang Weixu
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Zhao Chaoyue
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Lin Bin
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Song Shaojiang
(Department of Natural Products Chemistry, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)
Wang Shaojie
(Key Laboratory of Structure-Based Drugs Design & Discovery of Ministry of Education, School of Pharmaceutical Engineering, Shenyang Pharmaceutical University, 103 Culture Road, Shenhe District, Shenyang 110016, People’s Republic of China)

資料名:
European Journal of Medicinal Chemistry  (European Journal of Medicinal Chemistry)

巻: 138  ページ: 212-220  発行年: 2017年 
JST資料番号: E0845A  ISSN: 0223-5234  資料種別: 逐次刊行物 (A)
記事区分: 原著論文  発行国: オランダ (NLD)  言語: 英語 (EN)
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