文献
J-GLOBAL ID:201702258092498211
整理番号:17A0526841
独特なヒンジ結合を示す新しい,非常に強力なII型ABL/KIT二重キナーゼ阻害剤としての4-メチル-N-(4-((4-メチルピペラジン-1-イル)メチル)-3-(トリフルオロメチル)フェニル)-3-((1-ニコチノイルピペリジン-4-イル)オキシ)ベンズアミド(CHMFL-ABL/KIT-155)の発見
Discovery of 4-Methyl-N-(4-((4-methylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-3-((1-nicotinoylpiperidin-4-yl)oxy)benzamide (CHMFL-ABL/KIT-155) as a Novel Highly Potent Type II ABL/KIT Dual Kinase Inhibitor with a Distinct Hinge Binding
著者 (37件):
WANG Qiang
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Qiang
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
LIU Feiyang
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
LIU Feiyang
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
WANG Beilei
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Beilei
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
ZOU Fengming
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
ZOU Fengming
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
QI Ziping
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
QI Ziping
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
CHEN Cheng
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
CHEN Cheng
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
YU Kailin
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
YU Kailin
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
HU Chen
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
HU Chen
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
QI Shuang
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
QI Shuang
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
WANG Wenchao
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Wenchao
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
HU Zhenquan
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
HU Zhenquan
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
LIU Juan
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Wei
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Wei
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
WANG Li
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
WANG Li
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
LIANG Qianmao
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
ZHANG Shanchun
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
ZHANG Shanchun
(Hefei Cosource Medicine Technol. Co. Ltd., Anhui, CHN)
,
REN Tao
(Hefei Inst. of Physical Sci., Chinese Acad. of Sci., Anhui, CHN)
,
LIU Qingsong
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
LIU Qingsong
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
,
LIU Qingsong
(Univ. Sci. and Technol. of China, Anhui, CHN)
,
LIU Qingsong
(Hefei Inst. of Physical Sci., Chinese Acad. of Sci., Anhui, CHN)
,
LIU Jing
(High Magnetic Field Lab., Chinese Acad. of Sci., Anhui, CHN)
,
LIU Jing
(CHMFL-HCMTC Target Therapy Joint Lab., Anhui, CHN)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
60
号:
1
ページ:
273-289
発行年:
2017年01月12日
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)