文献
J-GLOBAL ID:201702291189589939
整理番号:17A0540131
全身曝露および前臨床データに基づくヒト中枢神経系における鎮静および非鎮静拮抗薬によるヒスタミンH1受容体占有率の定量的予測
Quantitative prediction of histamine H1 receptor occupancy by the sedative and non-sedative antagonists in the human central nervous system based on systemic exposure and preclinical data
著者 (6件):
Kanamitsu Kayoko
(Laboratory of Molecular Pharmacokinetics, Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo, 113-0033, Japan)
,
Kanamitsu Kayoko
(Tokushima Research Institute, Otsuka Pharmaceutical Co., Ltd., 463-10 Kagasuno, Kawauchi-cho, Tokushima-shi, Tokushima, 771-0192, Japan)
,
Nozaki Yoshitane
(Drug Metabolism and Pharmacokinetics Tsukuba, Tsukuba Research Laboratories, Eisai Co., Ltd., 5-1-3 Tokodai, Tsukuba-shi, Ibaraki, 300-2635, Japan)
,
Nagaya Yoko
(Drug Metabolism and Pharmacokinetics Tsukuba, Tsukuba Research Laboratories, Eisai Co., Ltd., 5-1-3 Tokodai, Tsukuba-shi, Ibaraki, 300-2635, Japan)
,
Sugiyama Yuichi
(Sugiyama Laboratory, RIKEN Innovation Center, Research Cluster for Innovation, RIKEN, 1-7-22 Suehiro-cho, Tsurumi-ku, Yokohama-shi, Kanagawa, 230-0045, Japan)
,
Kusuhara Hiroyuki
(Laboratory of Molecular Pharmacokinetics, Graduate School of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo, 113-0033, Japan)
資料名:
Drug Metabolism and Pharmacokinetics (Web)
(Drug Metabolism and Pharmacokinetics (Web))
巻:
32
号:
2
ページ:
135-144
発行年:
2017年04月
JST資料番号:
U0705A
ISSN:
1347-4367
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
オランダ (NLD)
言語:
英語 (EN)