文献
J-GLOBAL ID:201702291394166462
整理番号:17A0496846
BRD4阻害剤としての7-メチルイミダゾ[1,5-a]ピラジン-8(7H) -オン類似体の設計,合成および生物学的評価
Design, synthesis and biological evaluation of 7-methylimidazo[1,5-a]pyrazin-8(7H)-one derivatives as BRD4 inhibitors
著者 (7件):
Zhao Leilei
(Center of Drug Discovery, Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing 210009, PR China)
,
Yang Yifei
(Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China)
,
Guo Yahui
(Center of Drug Discovery, Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing 210009, PR China)
,
Yang Lingyun
(Center of Drug Discovery, Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing 210009, PR China)
,
Zhang Jian
(Center of Drug Discovery, Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing 210009, PR China)
,
Zhou Jinpei
(Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China)
,
Zhang Huibin
(Center of Drug Discovery, Jiangsu Key Laboratory of Drug Discovery for Metabolic Disease, China Pharmaceutical University, Nanjing 210009, PR China)
資料名:
Bioorganic & Medicinal Chemistry
(Bioorganic & Medicinal Chemistry)
巻:
25
号:
8
ページ:
2482-2490
発行年:
2017年04月15日
JST資料番号:
W0556A
ISSN:
0968-0896
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
オランダ (NLD)
言語:
英語 (EN)