文献
J-GLOBAL ID:201802217809763251
整理番号:18A0150681
pH依存性一般的塩基触媒活性化よりもむしろイソシアナート放流は関連1,2-ビス(メチルスルホニル)-1-(2-クロロエチル)ヒドラジンプロドラッグと比較したlaromustineの優れた抗腫瘍効果を説明するかもしれない【Powered by NICT】
pH-dependent general base catalyzed activation rather than isocyanate liberation may explain the superior anticancer efficacy of laromustine compared to related 1,2-bis(methylsulfonyl)-1-(2-chloroethyl)hydrazine prodrugs
著者 (6件):
Penketh Philip G.
(Department of Obstetrics, Gynecology & Reproductive Sciences, Yale University School of Medicine, New Haven, CT, USA)
,
Finch Richard A.
(Department of Veterinary Sciences, The University of Texas MD Anderson Cancer Center, Bastrop, TX, USA)
,
Sauro Rachel
(Department of Obstetrics, Gynecology & Reproductive Sciences, Yale University School of Medicine, New Haven, CT, USA)
,
Baumann Raymond P.
(Department of Pharmacology, Yale University School of Medicine, New Haven, CT, USA)
,
Ratner Elena S.
(Department of Obstetrics, Gynecology & Reproductive Sciences, Yale University School of Medicine, New Haven, CT, USA)
,
Shyam Krishnamurthy
(Department of Pharmacology, Yale University School of Medicine, New Haven, CT, USA)
資料名:
Chemical Biology & Drug Design
(Chemical Biology & Drug Design)
巻:
91
号:
1
ページ:
62-74
発行年:
2018年
JST資料番号:
A1436A
ISSN:
1747-0277
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)