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J-GLOBAL ID:201802259937087311   整理番号:18A0817790

ALPHALISAに基づくハイスループットスクリーニング分析による強力なDOT1L阻害剤の発見【JST・京大機械翻訳】

Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay
著者 (29件):
Song Yakai
(Nano Science and Technology Institute, University of Science and Technology of China, Suzhou 215123, China)
Song Yakai
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Li Linjuan
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Li Linjuan
(University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing 100049, China)
Li Linjuan
(School of Life Science and Technology, ShanghaiTech University, 100 Haike Road, Shanghai 201210, China)
Chen Yantao
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Chen Yantao
(University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing 100049, China)
Liu Jingqiu
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Liu Jingqiu
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Xiao Senhao
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Xiao Senhao
(University of Chinese Academy of Sciences, 19 Yuquan Road, Beijing 100049, China)
Xiao Senhao
(School of Life Science and Technology, ShanghaiTech University, 100 Haike Road, Shanghai 201210, China)
Lian Fulin
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Zhang Naixia
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Ding Hong
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Ding Hong
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Zhang Yuanyuan
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Zhang Yuanyuan
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Chen Kaixian
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Chen Kaixian
(Shanghai ChemPartner Co., Ltd., #5 Building, 998 Halei Road, Shanghai 201203, China)
Jiang Hualiang
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Jiang Hualiang
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Jiang Hualiang
(Shanghai ChemPartner Co., Ltd., #5 Building, 998 Halei Road, Shanghai 201203, China)
Zhang Chenhua
(Shanghai ChemPartner Co., Ltd., #5 Building, 998 Halei Road, Shanghai 201203, China)
Liu Yu-Chih
(Shanghai ChemPartner Co., Ltd., #5 Building, 998 Halei Road, Shanghai 201203, China)
Chen Shijie
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Chen Shijie
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Luo Cheng
(Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)
Luo Cheng
(CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China)

資料名:
Bioorganic & Medicinal Chemistry  (Bioorganic & Medicinal Chemistry)

巻: 26  号:ページ: 1751-1758  発行年: 2018年 
JST資料番号: W0556A  ISSN: 0968-0896  資料種別: 逐次刊行物 (A)
記事区分: 原著論文  発行国: オランダ (NLD)  言語: 英語 (EN)
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