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J-GLOBAL ID:201802268449937585   整理番号:18A0329544

ceritinibにおける末端ピペリジンの置換脂肪族アミンによるG1202R含むクリゾチニブ耐性変異株に対する活性を付与する【Powered by NICT】

Replacing the terminal piperidine in ceritinib with aliphatic amines confers activities against crizotinib-resistant mutants including G1202R
著者 (27件):
Mathi Gangadhar Rao
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Mathi Gangadhar Rao
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Kang Chung Hyo
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Kang Chung Hyo
(College of Pharmacy, Chungnam National University, Daejeon 34134, South Korea)
Lee Heung Kyoung
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Achary Raghavendra
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Achary Raghavendra
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Lee Ha-Yeon
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Lee Ha-Yeon
(College of Pharmacy, Chungbuk National University, Cheongju 28644, South Korea)
Lee Joo-Youn
(Korea Chemical Bank, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Ha Jae Du
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Ahn Sunjoo
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Ahn Sunjoo
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Park Chi Hoon
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Park Chi Hoon
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Lee Chong Ock
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Hwang Jong Yeon
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Hwang Jong Yeon
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Yun Chang-Soo
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Yun Chang-Soo
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Jung Hee Jung
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Jung Hee Jung
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Cho Sung Yun
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Cho Sung Yun
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)
Kim Hyoung Rae
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Kim Pilho
(Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 34114, South Korea)
Kim Pilho
(Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon 34113, South Korea)

資料名:
European Journal of Medicinal Chemistry  (European Journal of Medicinal Chemistry)

巻: 126  ページ: 536-549  発行年: 2017年 
JST資料番号: E0845A  ISSN: 0223-5234  資料種別: 逐次刊行物 (A)
記事区分: 原著論文  発行国: オランダ (NLD)  言語: 英語 (EN)
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