文献
J-GLOBAL ID:201902221847743720
整理番号:19A0176927
阻害剤と複合体を形成したERAP2の結晶構造は阻害剤の効力を最適化するための薬理作用団の必要性を明らか【JST・京大機械翻訳】
Crystal Structures of ERAP2 Complexed with Inhibitors Reveal Pharmacophore Requirements for Optimizing Inhibitor Potency
著者 (11件):
Mpakali Anastasia
(National Center for Scientific Research Demokritos, Greece)
,
Giastas Petros
(National Center for Scientific Research Demokritos, Greece)
,
Deprez-Poulain Rebecca
(Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs & Molecules for Living Systems, France)
,
Papakyriakou Athanasios
(National Center for Scientific Research Demokritos, Greece)
,
Koumantou Despoina
(National Center for Scientific Research Demokritos, Greece)
,
Gealageas Ronan
(Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs & Molecules for Living Systems, France)
,
Tsoukalidou Sofia
(National Center for Scientific Research Demokritos, Greece)
,
Vourloumis Dionisios
(National Center for Scientific Research Demokritos, Greece)
,
Mavridis Irene M.
(National Center for Scientific Research Demokritos, Greece)
,
Stratikos Efstratios
(National Center for Scientific Research Demokritos, Greece)
,
Saridakis Emmanuel
(National Center for Scientific Research Demokritos, Greece)
資料名:
ACS Medicinal Chemistry Letters
(ACS Medicinal Chemistry Letters)
巻:
8
号:
3
ページ:
333-337
発行年:
2017年
JST資料番号:
W5043A
ISSN:
1948-5875
資料種別:
逐次刊行物 (A)
記事区分:
短報
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)