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J-GLOBAL ID:201902238907869188   整理番号:19A0656270

乳酸デヒドロゲナーゼ(LDH)の強力な細胞活性ピラゾール系阻害剤の発見と最適化【JST・京大機械翻訳】

Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase (LDH)
著者 (29件):
Rai Ganesha
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Brimacombe Kyle R.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Mott Bryan T.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Urban Daniel J.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Hu Xin
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Yang Shyh-Ming
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Lee Tobie D.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Cheff Dorian M.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Kouznetsova Jennifer
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Benavides Gloria A.
(Mitochondrial Medicine Laboratory, Department of Pathology, University of Alabama at Birmingham, Alabama, United States)
Pohida Katie
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Kuenstner Eric J.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Luci Diane K.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Lukacs Christine M.
(Beryllium Discovery Corp., Washington, United States)
Davies Douglas R.
(Beryllium Discovery Corp., Washington, United States)
Dranow David M.
(Beryllium Discovery Corp., Washington, United States)
Zhu Hu
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Sulikowski Gary
(Vanderbilt Institute of Chemical Biology, Vanderbilt University, Tennessee, United States)
Moore William J.
(NExT Program Support, Applied/Developmental Research Directorate, Leidos Biomedical Research, Inc., Frederick National Laboratory for Cancer Research, Maryland, United States)
Stott Gordon M.
(NExT Program Support, Applied/Developmental Research Directorate, Leidos Biomedical Research, Inc., Frederick National Laboratory for Cancer Research, Maryland, United States)
Flint Andrew J.
(NExT Program Support, Applied/Developmental Research Directorate, Leidos Biomedical Research, Inc., Frederick National Laboratory for Cancer Research, Maryland, United States)
Hall Matthew D.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Darley-Usmar Victor M.
(Mitochondrial Medicine Laboratory, Department of Pathology, University of Alabama at Birmingham, Alabama, United States)
Neckers Leonard M.
(Urologic Oncology Branch, Center for Cancer Research, National Cancer Institute, Maryland, United States)
Dang Chi V.
(Abramson Cancer Center, Abramson Family Cancer Research Institute, Perelman School of Medicine, University of Pennsylvania, Pennsylvania, United States)
Waterson Alex G.
(Vanderbilt Institute of Chemical Biology, Vanderbilt University, Tennessee, United States)
Simeonov Anton
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Jadhav Ajit
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)
Maloney David J.
(National Center for Advancing Translational Sciences, National Institutes of Health, Maryland, United States)

資料名:
Journal of Medicinal Chemistry  (Journal of Medicinal Chemistry)

巻: 60  号: 22  ページ: 9184-9204  発行年: 2017年 
JST資料番号: D0102A  ISSN: 0022-2623  CODEN: JMCMAR  資料種別: 逐次刊行物 (A)
記事区分: 原著論文  発行国: アメリカ合衆国 (USA)  言語: 英語 (EN)
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