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J-GLOBAL ID:201902269360881881   整理番号:19A0176836

一連のピラゾロ[1,5-a]ピリミジン類から誘導されたCNS penetrant MGlu_7/8受容体PAM,VU60649の発見【JST・京大機械翻訳】

Discovery of VU6005649, a CNS Penetrant mGlu7/8 Receptor PAM Derived from a Series of Pyrazolo[1,5-a]pyrimidines
著者 (35件):
Abe Masahito
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Abe Masahito
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Seto Mabel
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Seto Mabel
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Gogliotti Rocco G.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Gogliotti Rocco G.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Loch Matthew T.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Loch Matthew T.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Bollinger Katrina A.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Chang Sichen
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Engelberg Eileen M.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Engelberg Eileen M.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Luscombe Vincent B.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Luscombe Vincent B.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Harp Joel M.
(Department of Biochemistry, Vanderbilt University School of Medicine, Tennessee, United States)
Bubser Michael
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Bubser Michael
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Engers Darren W.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Engers Darren W.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Jones Carrie K.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Jones Carrie K.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Jones Carrie K.
(Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Tennessee, United States)
Rodriguez Alice L.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Rodriguez Alice L.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Blobaum Anna L.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Blobaum Anna L.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Conn P. Jeffrey
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Conn P. Jeffrey
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Conn P. Jeffrey
(Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Tennessee, United States)
Niswender Colleen M.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Niswender Colleen M.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Niswender Colleen M.
(Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Tennessee, United States)
Lindsley Craig W.
(Department of Pharmacology, Vanderbilt University School of Medicine, Tennessee, United States)
Lindsley Craig W.
(Vanderbilt Center for Neuroscience Drug Discovery, Vanderbilt University School of Medicine, Tennessee, United States)
Lindsley Craig W.
(Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Tennessee, United States)

資料名:
ACS Medicinal Chemistry Letters  (ACS Medicinal Chemistry Letters)

巻:号: 10  ページ: 1110-1115  発行年: 2017年 
JST資料番号: W5043A  ISSN: 1948-5875  資料種別: 逐次刊行物 (A)
記事区分: 短報  発行国: アメリカ合衆国 (USA)  言語: 英語 (EN)
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