文献
J-GLOBAL ID:201902290146621480
整理番号:19A0656262
5-((5-([1,1′-ビフェニル]-4-イル)-6-クロロ-1H-ベンゾ[d]イミダゾール-2-イル)オキシ)-2-メチル安息香酸(MK-3903))のヒットからリードまでの最適化と発見:AMP活性化蛋白質キナーゼの新しいクラスのベンゾイミダゾールに基づく活性化剤【JST・京大機械翻訳】
Hit-to-Lead Optimization and Discovery of 5-((5-([1,1′-Biphenyl]-4-yl)-6-chloro-1H-benzo[d]imidazol-2-yl)oxy)-2-methylbenzoic Acid (MK-3903): A Novel Class of Benzimidazole-Based Activators of AMP-Activated Protein Kinase
著者 (23件):
Lan Ping
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Romero F. Anthony
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Wodka Dariusz
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Kassick Andrew J.
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Dang Qun
(Metabasis Therapeutics, Inc., La Jolla, United States)
,
Gibson Tony
(Metabasis Therapeutics, Inc., La Jolla, United States)
,
Cashion Daniel
(Metabasis Therapeutics, Inc., La Jolla, United States)
,
Zhou Gaochao
(Department of Biology, Merck & Co., Inc.)
,
Chen Yuli
(Department of Biology, Merck & Co., Inc.)
,
Zhang Xiaoping
(Department of Biology, Merck & Co., Inc.)
,
Zhang Aihua
(Department of Biology, Merck & Co., Inc.)
,
Li Ying
(Department of Biology, Merck & Co., Inc.)
,
Trujillo Maria E.
(Department of Pharmacology, Merck & Co., Inc.)
,
Shao Qing
(Department of Pharmacology, Merck & Co., Inc.)
,
Wu Margaret
(Department of Pharmacology, Merck & Co., Inc.)
,
Xu Shiyao
(Department of Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, MRL, Merck & Co., Inc.)
,
He Huaibing
(Department of Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, MRL, Merck & Co., Inc.)
,
MacKenna Deidre
(Metabasis Therapeutics, Inc., La Jolla, United States)
,
Staunton Jocelyn
(Metabasis Therapeutics, Inc., La Jolla, United States)
,
Chapman Kevin T.
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Weber Ann
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Sebhat Iyassu K.
(Department of Medicinal Chemistry, Merck & Co., Inc.)
,
Makara Gergely M.
(Department of Medicinal Chemistry, Merck & Co., Inc.)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
60
号:
21
ページ:
9040-9052
発行年:
2017年
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)