文献
J-GLOBAL ID:202002246251478410
整理番号:20A0427664
ジヒドロイソキノリノン二環コアを含む強力で選択的なWD反復ドメイン5(WDR5)阻害剤の発見と構造に基づく最適化【JST・京大機械翻訳】
Discovery and Structure-Based Optimization of Potent and Selective WD Repeat Domain 5 (WDR5) Inhibitors Containing a Dihydroisoquinolinone Bicyclic Core
著者 (30件):
Tian Jianhua
(Chemical Synthesis Core, Vanderbilt Institute of Chemical Biology, Vanderbilt University)
,
Teuscher Kevin B.
(Department of Biochemistry, Vanderbilt University)
,
Aho Erin R.
(Department of Cell and Developmental Biology, Vanderbilt University)
,
Alvarado Joseph R.
(Department of Biochemistry, Vanderbilt University)
,
Mills Jonathan J.
(Department of Biochemistry, Vanderbilt University)
,
Meyers Kenneth M.
(Department of Biochemistry, Vanderbilt University)
,
Gogliotti Rocco D.
(Department of Biochemistry, Vanderbilt University)
,
Han Changho
(Department of Biochemistry, Vanderbilt University)
,
Macdonald Jonathan D.
(Department of Biochemistry, Vanderbilt University)
,
Sai Jiqing
(Department of Biochemistry, Vanderbilt University)
,
Shaw J. Grace
(Department of Biochemistry, Vanderbilt University)
,
Sensintaffar John L.
(Department of Biochemistry, Vanderbilt University)
,
Zhao Bin
(Department of Biochemistry, Vanderbilt University)
,
Rietz Tyson A.
(Department of Biochemistry, Vanderbilt University)
,
Thomas Lance R.
(Department of Cell and Developmental Biology, Vanderbilt University)
,
Payne William G.
(Department of Biochemistry, Vanderbilt University)
,
Moore William J.
(Leidos Biomedical Research, Frederick National Laboratory for Cancer Research, Maryland, United States)
,
Stott Gordon M.
(Leidos Biomedical Research, Frederick National Laboratory for Cancer Research, Maryland, United States)
,
Kondo Jumpei
(Department of Clinical Bio-Resource Research and Development, Graduate School of Medicine, Kyoto University, Japan)
,
Kondo Jumpei
(Department of Biochemistry, Osaka International Cancer Institute, Japan)
,
Inoue Masahiro
(Department of Clinical Bio-Resource Research and Development, Graduate School of Medicine, Kyoto University, Japan)
,
Inoue Masahiro
(Department of Biochemistry, Osaka International Cancer Institute, Japan)
,
Coffey Robert J.
(Department of Cell and Developmental Biology, Vanderbilt University)
,
Coffey Robert J.
(Department of Medicine, School of Medicine, Vanderbilt University)
,
Tansey William P.
(Department of Cell and Developmental Biology, Vanderbilt University)
,
Stauffer Shaun R.
(Department of Biochemistry, Vanderbilt University)
,
Lee Taekyu
(Department of Biochemistry, Vanderbilt University)
,
Fesik Stephen W.
(Department of Biochemistry, Vanderbilt University)
,
Fesik Stephen W.
(Department of Pharmacology, Vanderbilt University)
,
Fesik Stephen W.
(Department of Chemistry, Vanderbilt University)
資料名:
Journal of Medicinal Chemistry
(Journal of Medicinal Chemistry)
巻:
63
号:
2
ページ:
656-675
発行年:
2020年
JST資料番号:
D0102A
ISSN:
0022-2623
CODEN:
JMCMAR
資料種別:
逐次刊行物 (A)
記事区分:
原著論文
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)