文献
J-GLOBAL ID:202202266644900470
整理番号:22A0726595
2つのS_NAr反応,酸化およびSuzukiカップリングを含む二重ロイシンジッパーキナーゼ阻害剤GDC-0134のための実用的およびよりグリーンなプロセスの開発【JST・京大機械翻訳】
Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two SNAr Reactions, Oxidation and Suzuki Coupling
著者 (15件):
Hoffmann-Emery Fabienne
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Niedermann Katrin
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Rege Pankaj D.
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Konrath Manuel
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Lautz Christian
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Kraft Anne Katrin
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Steiner Carine
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Bliss Fritz
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Hell Andre
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Fischer Rolf
(Synthetic Molecules Technical Development, F. Hoffmann-la Roche Ltd., Switzerland)
,
Carrera Diane E.
(Department of Small Molecule Process Chemistry, Genentech Inc., California, United States)
,
Beaudry Danial
(Department of Small Molecule Process Chemistry, Genentech Inc., California, United States)
,
Angelaud Remy
(Department of Small Molecule Process Chemistry, Genentech Inc., California, United States)
,
Malhotra Sushant
(Department of Small Molecule Process Chemistry, Genentech Inc., California, United States)
,
Gosselin Francis
(Department of Small Molecule Process Chemistry, Genentech Inc., California, United States)
資料名:
Organic Process Research & Development
(Organic Process Research & Development)
巻:
26
号:
2
ページ:
313-322
発行年:
2022年
JST資料番号:
W1013A
ISSN:
1083-6160
CODEN:
OPRDFK
資料種別:
逐次刊行物 (A)
記事区分:
文献レビュー
発行国:
アメリカ合衆国 (USA)
言語:
英語 (EN)