研究者
J-GLOBAL ID:201801005666935519   更新日: 2024年06月23日

増野 弘幸

マスノ ヒロユキ | Masuno Hiroyuki
所属機関・部署:
職名: 技術専門職員
研究分野 (1件): 薬系化学、創薬科学
競争的資金等の研究課題 (3件):
  • 2015 - 2018 新規ビタミンD受容体リガンドを目指した胆汁酸誘導体の構造活性相関研究
  • 2006 - 2008 エイズ・癌・慢性関節リウマチ等の難治性疾患に対するペプチド創薬研究
  • 2006 - 2007 胆汁酸誘導体のビタミンD受容体アゴニスト活性の構造生物学的解析
論文 (33件):
  • Ryosuke Ishida, Nagomi Kurebayashi, Hiroto Iinuma, Xi Zeng, Shuichi Mori, Masami Kodama, Takashi Murayama, Hiroyuki Masuno, Fumi Takeda, Masatoshi Kawahata, et al. A potent and selective cis-amide inhibitor of ryanodine receptor 2 as a candidate for cardiac arrhythmia treatment. European Journal of Medicinal Chemistry. 2023. 262. 115910-115910
  • Shigeru Yamada, Hiroyuki Masuno, Hiroyuki Kagechika, Aya Tanatani, Yasunari Kanda. A Novel Lithocholic Acid Derivative Upregulates Detoxification-Related Genes in Human Induced Pluripotent Stem Cell-Derived Intestinal Organoids. BIOLOGICAL & PHARMACEUTICAL BULLETIN. 2022. 45. 11. 1720-1724
  • Tsuyoshi Oikawa, Shinya Fujii, Shuichi Mori, Hiroyuki Masuno, Emiko Kawachi, Hiroyuki Kagechika. Structural Development of Silicon-Containing Retinoids: Structure-Activity Relationship Study of the Hydrophobic Pharmacophore of Retinobenzoic Acids Using Silyl Functionalities. CHEMMEDCHEM. 2022. 17. 12
  • Ayana Yoshihara, Haru Kawasaki, Hiroyuki Masuno, Koki Takada, Nobutaka Numoto, Nobutoshi Ito, Naoya Hirata, Yasunari Kanda, Michiyasu Ishizawa, Makoto Makishima, et al. Lithocholic Acid Amides as Potent Vitamin D Receptor Agonists. BIOMOLECULES. 2022. 12. 1
  • Shinya Fujii, Eriko Kikuchi, Honoka Suzuyama, Yuko Watanabe, Mari Ishigami-Yuasa, Hiroyuki Masuno, Takayasu Mori, Kiyoshi Isobe, Shinichi Uchida, Hiroyuki Kagechika. Structural Development of Salicylanilide-Based SPAK Inhibitors as Candidate Antihypertensive Agents. CHEMMEDCHEM. 2021. 16. 18. 2817-2822
もっと見る
MISC (1件):
  • K Yamamoto, H Masuno, S Yamada. Three-dimensional structure-activity relationship of vitamin D based on computational and synthetic chemistries. JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN. 2001. 59. 2. 131-141
特許 (5件):
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