Rchr
J-GLOBAL ID：200901073375398520
Update date: Feb. 14, 2024
Tarui Atsushi
タルイ アツシ | Tarui Atsushi
Affiliation and department：
Job title：
Lecturer
Homepage URL (1)：
http://www.setsunan.ac.jp/
Research field (3)：
Pharmaceuticals - chemistry and drug development
, Bioorganic chemistry
, Structural/physical organic chemistry
Research theme for competitive and other funds (2)：
- 2016 - 2017 フッ素化ペプチドの立体的相互作用を解析するための生化学ツールとなるフッ素化ペプチドの合成
- 2006 - 有機フッ素化合物の新規合成法の開発とその応用
Papers (68)：
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Yukiko Karuo, Atushi Tarui, Kazuyuki Sato, Kentaro Kawai, Masaaki Omote. Reactions Using Freons and Halothane as Halofluoroalkyl/Halofluoroalkenyl Building Blocks. The Chemical Record. 2023
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Motoyuki Isoda, Kazuyuki Sato, Kenta Kameda, Kana Wakabayashi, Ryota Sato, Hideki Minami, Yukiko Karuo, Atsushi Tarui, Kentaro Kawai, Masaaki Omote. Rhodium-catalyzed intramolecular reductive aldol-type cyclization: Application for the synthesis of a chiral necic acid lactone. Beilstein Journal of Organic Chemistry. 2022. 18. 1642-1648
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Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Kentaro Kawai, Masaaki Omote. Simple synthesis of multi-halogenated alkenes from 2-bromo-2-chloro-1,1,1-trifluoroethane (halothane). Beilstein Journal of Organic Chemistry. 2022. 18. 1567-1574
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Susumu Shinya, Kentaro Kawai, Naoki Kobayashi, Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Masato Otsuka, Masaaki Omote. Fluorophenylalkyl-substituted cyanoguanidine derivatives as bacteria-selective MATE transporter inhibitors for the treatment of antibiotic-resistant infections. Bioorganic & Medicinal Chemistry. 2022. 74. 117042-117042
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Kentaro Kawai, Jun Okada, Mizuki Nakae, Toshiki Tsujimura, Yukiko Karuo, Atsushi Tarui, Kazuyuki Sato, Shinji Yamashita, Makoto Kataoka, Masaaki Omote. Discovery of benzyloxyphenyl- and phenethylphenyl-imidazole derivatives as a new class of ante-drug type boosters. Bioorganic & Medicinal Chemistry Letters. 2022. 72. 128868-128868
ｍore...
MISC (2)：
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Atsushi Tarui, Kazuyuki Sato, Masaaki Omote, Itsumaro Kumadaki, Akira Ando. Stereoselective Synthesis of alpha-Fluorinated Amino Acid Derivatives. ADVANCED SYNTHESIS & CATALYSIS. 2010. 352. 16. 2733-2744
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K Sato, A Tarui, T Kita, Y Ishida, H Tamura, M Omote, A Ando, Kumadaki, I. Rhodium-catalyzed Reformatsky-type reaction of ethyl bromodifluoroacetate (vol 45, pg 5735, 2004). TETRAHEDRON LETTERS. 2005. 46. 5. 895-895
Books (1)：
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フッ素化学入門2015 フッ素化合物の合成法
三共出版 2015 ISBN:9784782707272
Lectures and oral presentations (245)：
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フッ素置換キノリン合成のためのカスケード型反応における反応機構解析へのアプローチ
(日本薬学会第143年会 2023)
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Krapcho脱炭酸を鍵とした連続反応による含フッ素キノリン合成法の開発
(日本薬学会関西支部大会 2022)
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プロテアーゼ阻害剤シード化合物となるフッ素化ジペプチドの酵素的速度論的分割とその活性
(日本薬学会関西支部大会 2022)
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機能性分子を指向したフッ素化-β-ラクタムの構造変換
(第42回有機合成若手セミナー 2022)
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Yb(OTf)3·nH2O accelerated cascade reaction of Krapcho decarboxylation and aldol reaction for the synthesis of α,α-difluoro-β-hydroxy ketones and its related compounds
(2021)
ｍore...
Education (3)：
- - 2006 Setsunan University Graduate School, Division of Pharmaceutical Sciences
- - 2006 Setsunan University Graduate School, Division of Pharmaceutical Sciences
- - 2004 Setsunan University Faculty of Pharmaceutical Science
Professional career (3)：
- B.S. (Pharmaceutical Sciences) (Setsunan University)
- M.S. (Pharmaceutical Sciences) (Setsunan University)
- Ph. D (Pharmaceutical Sciences) (Setsunan University)
Awards (1)：
- 2015/01 - 日本薬学会近畿支部 日本薬学会近畿支部奨励賞
Association Membership(s) (4)：
有機合成化学協会
, 日本フッ素化学会
, 日本薬学会
, American Chemical Society
