Art

J-GLOBAL ID：200902176592776220   Reference number：02A0433023

Peptidotriazoles on Solid Phase: [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides.

固相上のペプチドトリアゾール 銅(I)を触媒とした位置特異的な末端アルキンに対するアジドの1,3-双極性環状付加による[1,2,3]-トリアゾールの合成

Author (3)： TORNOE C W (Carlsberg Lab., Valby, DNK) ,  CHRISTENSEN C (Carlsberg Lab., Valby, DNK) ,  MELDAL M (Carlsberg Lab., Valby, DNK)
Material： Journal of Organic Chemistry  (J Org Chem)
Volume： 67  Issue： 9  Page： 3057-3064  Publication year： May. 03, 2002 
JST Material Number： C0328A  ISSN： 0022-3263  CODEN： JOCEAH  Document type： Article
Article type： 原著論文  Country of issue： United States (USA)  Language： ENGLISH (EN)

Thesaurus term： solid phase polymerization ,...

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JST classification (2)： Peptides  (CF10080G) ,  Triazoles  (CF07084O)

Substance index (36)： N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylpropyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-ethylpropyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-propylbutyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(Carboxydiphenylmethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(Carboxymethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxypentyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxypentadecyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(α-Carboxybenzyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(4-Aminophenyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-[(S)-2-Amino-5-guanidinopentyl]-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-[(S)-2-Amino-3-carboxypropyl]-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(2-Aminoethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-[(S)-2-Amino-4-(methylthio)butyl]-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-[(S)-2-Amino-3-phenylpropyl]-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Adamantyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Phenyl-2-deoxy-1-thio-α-D-galactopyranose-2-yl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-Phe-Gly-OH ester ,  N-(1H-1,2,3-Triazole-4-ylcarbonyl)-Phe-Gly-Phe-Gly-OH ,  3-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-yl]-Ala-Phe-Gly-Phe-Gly-OH ,  3-[1-(1-Phenyl-2-deoxy-1-thio-α-D-galactopyranose-2-yl)-1H-1,2,3-triazole-4-yl]-Ala-Phe-Gly-Phe-Gly-OH ester ,  3-[1-(4-Aminophenyl)-1H-1,2,3-triazole-4-yl]-Ala-Phe-Gly-Phe-Gly-OH ,  3-[1-[(S)-2-Benzyl-2-(Fmoc-amino)ethyl]-1H-1,2,3-triazole-4-yl]-Ala-Phe-Gly-Phe-Gly-OH ,  3-(1H-1,2,3-Triazole-4-yl)-Ala-Phe-Gly-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-OH ,  N-[1-(1-Adamantyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Ala-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Pro-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-O-tert-butyl-Thr-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-O-tert-butyl-Tyr-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-3-Boc-Ala-Phe-Gly-OH ,  N²-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-N⁴-trityl-Asn-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-1-trityl-His-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-S-trityl-Cys-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-Met-Phe-Gly-OH ,  N²-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-N⁶-Boc-Lys-Phe-Gly-OH ,  N-[1-(1-Carboxy-1-methylethyl)-1H-1,2,3-triazole-4-ylcarbonyl]-1-Boc-Trp-Phe-Gly-OH

Terms in the title (7)： 固相 ,  銅 ,  触媒 ,  末端アルキン ,  アジド ,  環状付加 ,  トリアゾール