Art

J-GLOBAL ID：200902194696748340   Reference number：01A1036336

Novel synthesis of tetrahydro-2(1H)-quinolones using Diels-Alder reactions of 1-arylsulfonyl-2(1H)-pyridones having an electron-withdrawing group.

電子求引基を有する1-アリールスルホニル-2(1H)-ピリドン類のDiels-Alder反応を用いるテトラヒドロ-2(1H)-キノロン類の新規な合成

Author (7)： FUJITA R (Tohoku Pharmaceutical Univ., Sendai, JPN) ,  WATANABE K (Tohoku Pharmaceutical Univ., Sendai, JPN) ,  IKEURA W (Tohoku Pharmaceutical Univ., Sendai, JPN) ,  OHTAKE Y (Tohoku Pharmaceutical Univ., Sendai, JPN) ,  HONGO H (Tohoku Pharmaceutical Univ., Sendai, JPN) ,  HARIGAYA Y (Kitasato Univ. Pharmaceutical Sci., Tokyo, JPN) ,  MATSUZAKI H (Tohoku Pharmaceutical Univ., Sendai, JPN)
Material： Tetrahedron  (Tetrahedron Symposia-in-Print)
Volume： 57  Issue： 42  Page： 8841-8850  Publication year： Oct. 15, 2001 
JST Material Number： E0234A  ISSN： 0040-4020  Document type： Article
Article type： 原著論文  Country of issue： United Kingdom (GBR)  Language： ENGLISH (EN)

Thesaurus term： Diels-Alder reaction ,...

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JST classification (1)： Quinolines,isoquinolines  (CF07096H)

Substance index (48)： 2-Oxo-1,2-dihydropyridine-5-carboxylic acid methyl ester ,  5-Acetylpyridine-2(1H)-one ,  5-Nitropyridin-2-ol ,  5-Bromo-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1,2-Dihydro-2-oxopyridine-4-carboxylic acid methyl ester ,  p-Toluenesulfonic acid chloride ,  4-Methoxybenzenesulfonic acid chloride ,  4-Chlorobenzenesulfonic acid chloride ,  4-Nitrobenzenesulfonic acid chloride ,  Benzenesulfonic acid chloride ,  o-Toluenesulfonyl chloride ,  2-Mesitylenesulfonyl chloride ,  2,4,6-Triisopropylbenzenesulfonyl chloride ,  6-[(2,4,6-Trimethylphenylsulfonyl)oxy]pyridine-3-carboxylic acid ,  1-Tosyl-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-Tosyl-5-acetyl-2(1H)-pyridone ,  1-Tosyl-5-nitro-2(1H)-pyridone ,  1-(4-Methoxyphenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(4-Chlorophenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(4-Nitrophenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(Phenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(2-Methylphenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(2,4,6-Trimethylphenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(2,4,6-Triisopropylphenylsulfonyl)-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(4-Methylphenylsulfonyl)-5-bromo-6-oxo-1,6-dihydropyridine-3-carboxylic acid methyl ester ,  1-(4-Methylphenylsulfonyl)-6-oxo-1,6-dihydropyridine-4-carboxylic acid methyl ester ,  6-[(2,4,6-Triisopropylphenylsulfonyl)oxy]pyridine-3-carboxylic acid ,  1-Tosyl-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  1-Tosyl-4aα-acetyl-6,7-dimethyl-4a,5,8,8aα-tetrahydroquinoline-2(1H)-one ,  1-Tosyl-4aα-nitro-6,7-dimethyl-4a,5,8,8aα-tetrahydroquinoline-2(1H)-one ,  1-[(4-Methoxyphenyl)sulfonyl]-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  1-[(4-Chlorophenyl)sulfonyl]-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  1-[(4-Nitrophenyl)sulfonyl]-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  1-(Phenylsulfonyl)-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  (4aS)-1-(2-Methylphenylsulfonyl)-2-oxo-6,7-dimethyl-1,2,4a,5,8,8aα-hexahydroquinoline-4aα-carboxylic acid methyl ester ,  1-[(2,4,6-Trimethylphenyl)sulfonyl]-2-oxo-6,7-dimethyl-1,2,8,8aα-tetrahydroquinoline-4aα(5H)-carboxylic acid methyl ester ,  (4aS)-1-(2,4,6-Triisopropylphenylsulfonyl)-2-oxo-6,7-dimethyl-1,2,4a,5,8,8aα-hexahydroquinoline-4aα-carboxylic acid methyl ester ,  (4aS)-1-(4-Methylphenylsulfonyl)-2-oxo-3-bromo-6,7-dimethyl-1,2,4a,5,8,8aα-hexahydroquinoline-4aα-carboxylic acid methyl ester ,  (4aS)-1-(4-Methylphenylsulfonyl)-2-oxo-3-bromo-7-methyl-1,2,4a,5,8,8aα-hexahydroquinoline-4aα-carboxylic acid methyl ester ,  6-[(4-Methylphenyl)sulfonyloxy]pyridine-3-carboxylic acid methyl ester ,  p-Toluenesulfonic acid 5-acetyl-2-pyridyl ester ,  6-[(4-Methoxyphenyl)sulfonyloxy]pyridine-3-carboxylic acid methyl ester ,  6-(Phenylsulfonyloxy)pyridine-3-carboxylic acid methyl ester ,  6-[(2-Methylphenylsulfonyl)oxy]-3-pyridinecarboxylic acid methyl ester ,  2,3-Dimethyl-1,3-butadiene ,  Isoprene ,  (4aS)-1-Oxo-2-(4-methylphenylsulfonyl)-6,7-dimethyl-1,2,4a,5,8,8aα-hexahydroisoquinoline-4aα-carboxylic acid methyl ester ,  (4aS)-1-Oxo-2-(4-methylphenylsulfonyl)-6,7-dimethyl-1,2,4a,5,8,8aβ-hexahydroisoquinoline-4aα-carboxylic acid methyl ester

Terms in the title (4)： 電子求引基 ,  ピリドン類 ,  Diels-Alder反応 ,  キノロン類