Art

J-GLOBAL ID：200902283081383352   Reference number：04A0415866

Synthesis of Chiral Sulfinyl-Substituted 1-Indolyl Enones and Asymmetric Conjugate Addition by an Arylcopper Reagent

キラルなスルフィニル置換1-インドリルエノン類の合成及びアリール銅試薬による不斉共役付加

Author (3)： ARAI Y (Gifu Pharmaceutical Univ., Gifu, JPN) ,  KASAI M (Gifu Pharmaceutical Univ., Gifu, JPN) ,  MASAKI Y (Gifu Pharmaceutical Univ., Gifu, JPN)
Material： Chemical and Pharmaceutical Bulletin  (Chemical & Pharmaceutical Bulletin)
Volume： 52  Issue： 6  Page： 733-738  Publication year： Jun. 01, 2004 
JST Material Number： G0504A  ISSN： 0009-2363  CODEN： CPBTAL  Document type： Article
Article type： 原著論文  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： *nitrogen heterocyclic compound ,...

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JST classification (2)： Condensed derivatives of pyrroles  (CF07077C) ,  Addition reaction,elimination reaction  (CF02030M)

Substance index (15)： (E)-1-[2-(p-Tolylsulfinyl)-1H-pyrrol-1-yl]-3-phenyl-2-propen-1-one ,  (E)-1-[2-(p-Tolylsulfinyl)-1H-pyrrole-1-yl]-3-phenyl-2-butene-1-one ,  2-(p-Tolylsulfinyl)-1H-pyrrole ,  (E)-1-[3-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-2-propene-1-one ,  (E)-1-[3-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-2-butene-1-one ,  (E)-1-[2-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-2-propene-1-one ,  (E)-1-[2-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-2-butene-1-one ,  1H-Indole-1-yl p-tolyl sulfoxide ,  1-Tosyl-3-iodo-1H-indole ,  Andersen reagent ,  3-(p-Tolylsulfinyl)-1H-indole-1-yl p-tolyl sulfone ,  (3S)-1-[3-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-3-p-tolyl-1-propanone ,  (3R)-1-[3-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-p-tolyl-1-butanone ,  (3R)-1-[2-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-phenyl-3-p-tolyl-1-propanone ,  (3S)-1-[2-(p-Tolylsulfinyl)-1H-indole-1-yl]-3-p-tolyl-1-butanone

Reference (15)：

• 1) Arai Y., Ueda K., Xie J., Masaki Y., Chem. Pharm. Bull., 49, 1609—1614 (2001).
• 2) Matsuzono M., Fukuda T., Iwao M., Tetrahedron Lett., 42, 7621—7623 (2001).
• 3) Kondo Y., Yoshida A., Sato S., Sakamoto T., Heterocycles, 42, 105—108 (1996).
• 4) Kano S., Sugino E., Shibuya S., Hibino S., J. Org. Chem., 46, 2979—2981 (1981).
• 5) Sailnier M. G., Gribble G. W., J. Org. Chem., 47, 757—761 (1982).

Terms in the title (5)： キラル ,  置換 ,  銅 ,  試薬 ,  共役付加