Art

J-GLOBAL ID：201102246061301924   Reference number：11A0945082

Affinity to the Nicotinic Acetylcholine Receptor and Insecticidal Activity of Chiral Imidacloprid Derivatives with a Methylated Imidazolidine Ring

メチル化イミダゾリジン環を持つキラルイミダクロプリド誘導体のニコチン性アセチルコリン受容体への親和性および殺虫活性

Author (5)： NISHIWAKI Hisashi (Fac. of Agriculture, Ehime Univ.) ,  NAGAOKA Hikaru (Fac. of Agriculture, Ehime Univ.) ,  KURIYAMA Mituhiro (Fac. of Agriculture, Ehime Univ.) ,  YAMAUCHI Satoshi (Fac. of Agriculture, Ehime Univ.) ,  SHUTO Yoshihiro (Fac. of Agriculture, Ehime Univ.)
Material： Bioscience, Biotechnology, and Biochemistry  (Bioscience Biotechnology & Biochemistry)
Volume： 75  Issue： 4  Page： 780-782 (J-STAGE)  Publication year： 2011 
JST Material Number： G0021A  ISSN： 0916-8451  CODEN： BBBIEJ  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： *nicotinic receptor ,  Musca domestica ,  *insecticidal action ,  single donor oxygenase ,  nitrogen heterocyclic compound ,  methylation ,  chemical synthesis ,  structure-activity relationship ,  synergism ,  organochlorine compound ,  nitramine
Semi thesaurus term： Imidazolidines ,  oxygenase ,  *nicotinic acetylcholine receptor ,  insecticidal activity

JST classification (1)： Pesticides to insect pest  (FB06020U)

Substance index (6)： Imidacloprid ,  1-(6-Chloro-3-pyridyl)-2-nitromethyleneimidazolidine ,  5-[(4R)-4-Methyl-2-(nitromethylene)-3-imidazolidinyl]-2-chloropyridine ,  5-[(5R)-5-Methyl-2-(nitromethylene)-3-imidazolidinyl]-2-chloropyridine ,  5-[(4S)-4-Methyl-2-(nitromethylene)-3-imidazolidinyl]-2-chloropyridine ,  5-[(5S)-5-Methyl-2-(nitromethylene)-3-imidazolidinyl]-2-chloropyridine

Reference (15)：

• 1) Elbert A, Overbeck H, Iwaya K, and Tsuboi S, “Proc Brighton Crop Protect Conf—Pests & Diseases,” BCPC, Farnham, pp. 21–28 (1990).
• 2) Kagabu S, J. Agric. Food Chem., 59, 2887–2896 (2011).
• 3) Sun C, Yang D, Xing J, Wang H, Jin J, and Zhu J, J. Agric. Food Chem., 58, 3415–3421 (2010).
• 4) Nishiwaki H, Nakagawa Y, Takeda DY, Okazawa A, Akamatsu M, Miyagawa H, Ueno T, and Nishimura K, Pest Manag. Sci., 56, 875–881 (2000).
• 5) Nishiwaki H, Nakagawa Y, Ueno T, Kagabu S, and Nishimura K, Pest Manag. Sci., 57, 810–814 (2001).

Terms in the title (7)： メチル化 ,  イミダゾリジン ,  環 ,  誘導体 ,  ニコチン性アセチルコリン受容体 ,  親和性 ,  殺虫活性