Art

J-GLOBAL ID：201302241554206192   Reference number：13A0316948

Novel synthesis of 1,4,5-trisubstituted 1,2,3-triazoles via a one-pot three-component reaction of boronic acids, azide, and active methylene ketones

ボロン酸,アジドおよび活性メチレンケトンのワンポット三成分反応による1,4,5-三置換1,2,3-トリアゾールの新規合成

Author (5)： ZHANG Jian (Shanghai Key Lab. of Chemical Biology, School of Pharmacy, East China Univ. of Sci. and Technol., Shanghai 200237, CHN) ,  JIN Guanyi (Shanghai Key Lab. of Chemical Biology, School of Pharmacy, East China Univ. of Sci. and Technol., Shanghai 200237, CHN) ,  XIAO Senhan (Shanghai Key Lab. of Chemical Biology, School of Pharmacy, East China Univ. of Sci. and Technol., Shanghai 200237, CHN) ,  WU Jingjing (Shanghai Key Lab. of Chemical Biology, School of Pharmacy, East China Univ. of Sci. and Technol., Shanghai 200237, CHN) ,  CAO Song (Shanghai Key Lab. of Chemical Biology, School of Pharmacy, East China Univ. of Sci. and Technol., Shanghai 200237, CHN)
Material： Tetrahedron  (Tetrahedron Symposia-in-Print)
Volume： 69  Issue： 10  Page： 2352-2356  Publication year： Mar. 11, 2013 
JST Material Number： E0234A  ISSN： 0040-4020  Document type： Article
Article type： 原著論文  Country of issue： United Kingdom (GBR)  Language： ENGLISH (EN)

Thesaurus term： *nitrogen heterocyclic compound ,  *chemical reaction ,  one-pot synthesis ,  azide(inorganic) ,  sodium compound ,  boron compound ,  organic compound
Semi thesaurus term： Sodium Azide ,  *Triazoles ,  Boronic acid ,  active methylene compound ,  *three-component reaction

JST classification (1)： Triazoles  (CF07084O)

Substance index (19)： 1,5-Diphenyl-1H-1,2,3-triazole-4-carbonitrile ,  1-Phenyl-4-acetyl-5-methyl-1H-1,2,3-triazole ,  1-(3-Nitrophenyl)-5-(trifluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Fluorophenyl)-5-(difluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Fluorophenyl)-5-(trifluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Fluorophenyl)-5-phenyl-1H-1,2,3-triazole-4-carbonitrile ,  1-(4-Methylphenyl)-5-(difluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Methylphenyl)-5-(trifluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Methoxyphenyl)-5-(difluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Methoxyphenyl)-5-(trifluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-(4-Methoxyphenyl)-5-phenyl-1H-1,2,3-triazole-4-carbonitrile ,  1-[1-(4-Methoxyphenyl)-5-methyl-1H-1,2,3-triazole-4-yl]ethanone ,  1-Phenyl-5-(difluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-Phenyl-5-(trifluoromethyl)-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  1-Phenyl-5-methyl-1H-1,2,3-triazole-4-carboxylic acid ethyl ester ,  Ethyl 4,4,4-trifluoroacetoacetate ,  Piperidine ,  Phenylboronic acid ,  Diacetic acid copper(II) salt

Terms in the title (7)： ボロン酸 ,  アジド ,  活性 ,  ポット ,  三成分反応 ,  置換 ,  トリアゾール