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J-GLOBAL ID：201602215555698481   Reference number：16A0154296

Synthesis and antibacterial activity of 4′′ or 6′′-alkanoylamino derivatives of arbekacin

アルベカシンの4′′または6′′-アルカノイルアミノ誘導体の合成と抗菌活性

Author (7)： SASAKI Kazushige (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  KOBAYASHI Yoshihiko (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  KURIHARA Takashi (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  YAMASHITA Yohei (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  TAKAHASHI Yoshiaki (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  MIYAKE Toshiaki (Inst. of Microbial Chemistry (BIKAKEN), Kawasaki, JPN) ,  AKAMATSU Yuzuru (Inst. of Microbial Chemistry (BIKAKEN), Tokyo, JPN)
Material： Journal of Antibiotics (Web)  (J Antibiot (Web))
Volume： 68  Issue： 12  Page： 741-747 (WEB ONLY)  Publication year： Dec. 2015 
JST Material Number： U0320A  ISSN： 0021-8820  Document type： Article
Article type： 原著論文  Country of issue： Germany, Federal Republic of (DEU)  Language： ENGLISH (EN)

Thesaurus term： *aminoglycoside antibiotics ,...
Semi thesaurus term： derivative

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JST classification (1)： Synthesis of antibiotics  (GX04000Z)

Substance index (1)： Arbekacin

Reference (26)：

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• Perez-Fernandez, D. et al. C. 4'-O-substitutions determine selectivity of aminoglycoside antibiotics. Nat. Commun. 5, 3112 (2014)
• Magnet, S. & Blanchard, S. Molecular insights into aminoglycoside action and resistance. J. Chem. Rev. 105, 477-498 (2005).

Terms in the title (3)： アルベカシン ,  誘導体 ,  抗菌活性