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J-GLOBAL ID：201602261575288834   Reference number：16A1175484

SYNTHESIS AND DNA CLEAVAGE ACTIVITY OF FUNCTIONALIZED PYRAZOL-3-ONES CONTAINING OXIME ESTER

官能化ピラゾール--3オン類含有オキシムエステルの合成およびDNA切断活性

Author (6)： MASUMOTO Eiichi (Fukuoka Univ., Fukuoka, JPN) ,  KASHIGE Nobuhiro (Fukuoka Univ., Fukuoka, JPN) ,  OKABE Fumi (Fukuoka Univ., Fukuoka, JPN) ,  MIAKE Fumio (Fukuoka Univ., Fukuoka, JPN) ,  YAMAGATA Kenji (Fukuoka Univ., Fukuoka, JPN) ,  MARUOKA Hiroshi (Fukuoka Univ., Fukuoka, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 92  Issue： 7  Page： 1293-1306  Publication year： Jul. 01, 2016 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： molecular genetic phenomenon ,...

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JST classification (2)： Pyrazoles  (CF07082G) ,  Molecular genetics in general  (EC02010J)

Substance index (10)： 4-[(E)-2-(Acetoxyimino)propyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(E)-2-(Propanoyloxyimino)propyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(E)-2-(Benzoyloxyimino)propyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(E)-2-(4-Nitrobenzoyloxyimino)propyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(E)-2-(4-Methoxybenzoyloxyimino)propyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(Z)-β-(Acetoxyimino)phenethyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(Z)-β-(Propanoyloxyimino)phenethyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(Z)-β-(Benzoyloxyimino)phenethyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(Z)-β-(4-Nitrobenzoyloxyimino)phenethyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one ,  4-[(Z)-β-(4-Methoxybenzoyloxyimino)phenethyl]-2-phenyl-4-hydroxy-5-methyl-2,4-dihydro-3H-pyrazole-3-one

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Terms in the title (5)： 官能化 ,  ピラゾール ,  オキシムエステル ,  DNA切断 ,  活性