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J-GLOBAL ID：201702212908197843   Reference number：17A0279699

FACILE AND CONVENIENT SYNTHESES OF FLUORINE-CONTAINING PYRIMIDO[5,4-c]QUINOLINES AND BENZO[h][1,6]NAPHTHYRIDINES BY CONDENSATION REACTION OF 2-METHOXY-3-TRIFLUOROACETYL-4-QUINOLYLAMINE WITH ALDEHYDES AND KETONES

2-メトキシ-3-トリフルオロアセチル-4-キノリルアミンとアルデヒドおよびケトンとの縮合反応によるフッ素含有ピリミド[5,4-c]キノリン類およびベンゾ[h][1,6]ナフチリジン類の簡易かつ簡便合成

Author (2)： HATAKENAKA Mizuki (Kobe Univ., Kobe, JPN) ,  OKADA Etsuji (Kobe Univ., Kobe, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 94  Issue： 1  Page： 102-116  Publication year： Jan. 01, 2017 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： nitrogen heterocyclic compound ,  polynuclear aromatic compound ,  chemical synthesis ,  *condensation reaction ,  aldehyde ,  ketone ,  organofluorine compound ,  chemical reaction
Semi thesaurus term： Quinolines ,  *Naphthyridines ,  *Pyrimidines ,  three-component reaction

JST classification (1)： Other condensed derivatives of pyridine  (CF07097Y)

Substance index (15)： 2-Methoxy-3-(trifluoroacetyl)-4-aminoquinoline ,  2-Methyl-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-Ethyl-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-Isopropyl-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-(4-Methoxyphenyl)-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-(4-Methylphenyl)-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-Phenyl-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  2-(4-Chlorophenyl)-4-(trifluoromethyl)-5-methoxy-1,2-dihydropyrimido[5,4-c]quinoline ,  9-Methyl-7-(trifluoromethyl)-6-methoxy-10-azabenzo[c]quinoline ,  8-Methyl-9-ethyl-7-(trifluoromethyl)-6-methoxy-10-azabenzo[c]quinoline ,  2-Ethyl-4-(trifluoromethyl)-5-methoxybenzo[h][1,6]naphthyridine ,  2-Isopropyl-4-(trifluoromethyl)-5-methoxybenzo[h][1,6]naphthyridine ,  9-Phenyl-7-(trifluoromethyl)-6-methoxy-10-azabenzo[c]quinoline ,  2,3-Trimethylene-4-(trifluoromethyl)-5-methoxybenzo[h][1,6]naphthyridine ,  6-Methoxy-7-(trifluoromethyl)-8,9,10,11-tetrahydrodibenzo[b,h][1,6]naphthyridine

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Terms in the title (8)： アルデヒド ,  ケトン ,  縮合反応 ,  フッ素 ,  キノリン類 ,  ナフチリジン類 ,  簡易 ,  簡便