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J-GLOBAL ID：202002250185123753   Reference number：20A0846383

SYNTHESIS AND BIOLOGICAL EVALUATION OF NMDI14 DERIVATIVES AS ANTI-MESOTHELIOMA AGENTS

抗中皮腫薬としてのNMDI14誘導体の合成と生物学的評価

Author (8)： NGUYEN Hong Nhung (Nagoya Univ., Aichi, JPN) ,  SUZUKI Koya (Juntendo Univ., Tokyo, JPN) ,  KIMURA Yasuaki (Nagoya Univ., Aichi, JPN) ,  HIROKAWA Takatsugu (AIST, Tokyo, JPN) ,  HIROKAWA Takatsugu (Univ. Tsukuba, Ibaraki, JPN) ,  MURAKAMI-TONAMI Yuko (Juntendo Univ., Tokyo, JPN) ,  ABE Hiroshi (Nagoya Univ., Aichi, JPN) ,  ABE Hiroshi (JST-CREST, Tokyo, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 100  Issue： 2  Page： 253-266  Publication year： Feb. 01, 2020 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： chemical synthesis ,...
Semi thesaurus term： mRNA decay ,...

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JST classification (2)： Pyrazines  (CF07104N) ,  Basic research of antitumor(=antineoplastic)drugs  (GW16010A)

Substance index (13)： 2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-(pyridin-2-yl)acetamide ,  2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-[(5-methylfuran-2-yl)methyl]acetamide ,  2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-(furan-2-ylmethyl)acetamide ,  2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-[2-(thiophen-2-yl)ethyl]acetamide ,  2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-phenylacetamide ,  2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)-N-propylacetamide ,  2-[6,7-dimethyl-1-(4-methylbenzenesulfonyl)-3-oxo-2,4-dihydroquinoxalin-2-yl]-N-propylacetamide ,  [6,7-dimethyl-1-(4-methylbenzenesulfonyl)-3-oxo-2,4-dihydroquinoxalin-2-yl]acetic acid ,  4,5-Dimethyl-o-phenylenediamine ,  NMDI-14 ,  ethyl 2-(6,7-dimethyl-3-oxo-2,4-dihydro-1H-quinoxalin-2-yl)acetate ,  ethyl 2-[(2E)-6,7-dimethyl-3-oxo-1,4-dihydroquinoxalin-2-ylidene]acetate ,  ethyl 2-[6,7-dimethyl-1-(4-methylbenzenesulfonyl)-3-oxo-2,4-dihydroquinoxalin-2-yl]acetate

Reference (11)：

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Terms in the title (3)： 中皮腫 ,  誘導体 ,  生物学的評価