【課題】ポロ様キナーゼ-1阻害効果を有する化合物またはその薬学的に許容し得る塩の提供。【解決手段】下記式[式中、Aで示される複素環は、ピリジン、ピリミジン、ジヒドロピリミジン、ベンゾイミダゾール、ベンゾチアゾール、ジヒドロチアゾール又はチアゾリジンを示し;Bで示される環は、ベンゼン又はフランを示し;R1はニトロ基、オキソ基、低級アルコキシ基、カルボキシル基、低級アルコキシカルボニル基、低級アルカノイル基、アミノ基、チオキソ基又はシアノ基を示し;R2はハロゲン原子、低級アルコキシ基、低級アルコキシカルボニル基、低級アルカノイル基又はシアノ基を示し;Xは-S-、-O-又は-NH-を示し;lは0〜3の整数を示し;mは0又は1の整数を示し;nは0〜3の整数を示し;pは0〜3の整数を示す]で表される複素環化合物又はその塩。【選択図】なし
出願人引用 (23件)
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1061903-99-8, 20081016
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 850375-95-0, 20050512
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 312266-71-0, 20001229
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 331421-74-0, 20010416
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 119022-84-3, 19890217
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 311809-92-4, 20011228
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 336181-11-4, 20010517
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 371205-06-0, 20011121
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 489414-10-0, 20030213
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-05-0, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-06-1, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-07-2, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-08-3, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-09-4, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-10-7, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-11-8, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-12-9, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-13-0, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-14-1, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-15-2, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-16-3, 20091027
全件表示
審査官引用 (23件)
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1061903-99-8, 20081016
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 850375-95-0, 20050512
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 680998-56-5, 20040510
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 893756-22-4, 20060717
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 312266-71-0, 20001229
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 331421-74-0, 20010416
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 119022-84-3, 19890217
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 311809-92-4, 20011228
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 336181-11-4, 20010517
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 371205-06-0, 20011121
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 489414-10-0, 20030213
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-05-0, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-06-1, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-07-2, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-08-3, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-09-4, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-10-7, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-11-8, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-12-9, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-13-0, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-14-1, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-15-2, 20091027
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REGISTRY (STN) [online] ; [retrieved on 22 Mar 2013],CAS Registry No. (RN): 1190205-16-3, 20091027
全件表示