Rchr
J-GLOBAL ID：200901074033822776   Update date: Oct. 10, 2024

Kitamura Yoshiaki

キタムラ ヨシアキ | Kitamura Yoshiaki
Affiliation and department：
Gifu University Faculty of Engineering

About Gifu University Faculty of Engineering


Other affiliations (4)：
  • Gifu University  Graduate School of Natural Science and Technology 
  • Gifu University  United Graduate School of Drug Discovery and Medical Information Sciences 
  • Gifu University  Center for One Medicine Innovative Translational Research 
  • Gifu University  Artificial Intelligence Advanced Research Center 
Homepage URL  (1)： https://www1.gifu-u.ac.jp/~kitam_rg/
Research field  (1)： Pharmaceuticals - chemistry and drug development
Research keywords  (8)： Synthesis of novel cancer imaging candidates ,  Transition metal catalyst ,  Molecular imaging ,  Nucleic acid chemistry ,  Organic synthesis ,  オリゴ核酸修飾 ,  核酸医薬 ,  siRNA
Research theme for competitive and other funds  (5)：
  • 2022 - 2025 Development of practical synthetic method for oligonucleotides
  • 2016 - 2018 Development of sophisticated small RNAs utilizing the properties of functional groups
  • 2012 - 2015 Owing to the development of RNA medicine, discovery of practical RNA molecules and synthesis of nucleic acid PET probes
  • 2010 - 2013 Novel modification method of oligonucleotides for siRNA medicine
  • 2011 - 2012 マイクロRNAの機能を利用した難治性疾患の早期診断法及び治療法の開発
Papers (69)：
  • Ryoga Sawahata, Yuga Takagi, Yoshiaki Kitamura. Azidomethylation of Nucleobases and Related N-Heterocycles, Benzazoles, and Bis(arene)sulfonimides Using Azidomethyl Esters with Silyl Triflates. Organic Letters. 2024. 26. 18. 3806-3809
  • Yoshiaki Kitamura, Mahmoud Kandeel, Erina Oba, Chiori Iwai, Keitaro Iritani, Nanako Nagaya, Reo Namura, Hiroshi Katagiri, Hiroshi Ueda, Yukio Kitade. A Diversifiable Synthetic Platform for the Discovery of New Carbasugar SGLT2 Inhibitors Using Azide-Alkyne Click Chemistry. Chemical and Pharmaceutical Bulletin. 2023. 71. 3. 240-249
  • Shintaro Sugiura, Yuki Shintani, Daisuke Mori, Sayuri L. Higashi, Aya Shibata, Yoshiaki Kitamura, Shin-ichiro Kawano, Koichiro M. Hirosawa, Kenichi G.N. Suzuki, Masato Ikeda. Design of supramolecular hybrid nanomaterials comprising peptide-based supramolecular nanofibers and in situ generated DNA nanoflowers through rolling circle amplification. Nanoscale. 2022. 15. 3. 1024-1031
  • Yuki Shintani, Taku Ohtomi, Aya Shibata, Yoshiaki Kitamura, Koichiro M. Hirosawa, Kenichi G. N. Suzuki, Masato Ikeda. Formation of Supramolecular Nanostructures through in Situ Self-Assembly and Post-Assembly Modification of a Biocatalytically Constructed Dipeptide Hydrazide**. Chemistry - A European Journal. 2022. 28. 8. e202104421
  • Yoshiaki Kitamura, Yuto Ohshima, Yuki Nagaya. A new approach for the synthesis of N-β-enaminocarbonyl 2-oxazolidinones through ring transformation reactions of uracil. Tetrahedron Letters. 2022. 88. 153554-153554
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MISC (11)：
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Patents (3)：
Books (3)：
  • 医薬品モダリティの 特許戦略と技術開発動向
    2019
  • Current Protocols in Nucleic Acid Chemistry
    2014
  • 固定化触媒のルネッサンス
    2007
Lectures and oral presentations  (166)：
  • アジドメチル化反応の開発と各種アミン類への適用
    (日本薬学会第144年会 2024)
  • 核酸オリゴマーの新規合成法の開発を指向した5’位官能基化チミジンモノマーの合成とリン酸ジエステルとの反応
    (日本薬学会第144年会 2024)
  • アジドメチルエステル類のアジドメチル化剤としての利用
    (第54回中部化学関係学協会支部連合秋季大会 2023)
  • 新規核酸オリゴマー構築法の開発を目指した5’位官能基化ヌクレオシド誘導体の合成
    (第49回反応と合成の進歩シンポジウム 2023)
  • フラノイドグリカールからフラン誘導体への変換を利用したプロドラッグ戦略
    (第49回反応と合成の進歩シンポジウム 2023)
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Works (1)：
  • 東海3大学新技術説明会
    2010 -
Education (3)：
  • 2006 - 2007 Gifu Pharmaceutical University Graduate School Department of Pharmaceutical Science
  • 2004 - 2006 Gifu Pharmaceutical University Graduate School Department of Pharmaceutical Science
  • 2000 - 2004 Gifu Pharmaceutical University Faculty of Pharmaceutical Science Department of Public Health Pharmacy
Professional career (1)：
  • 博士(薬学) (岐阜薬科大学)
Work history (7)：
  • 2023/09 - 現在 Gifu University
  • 2023/01 - 現在 Gifu University Center for One Medicine Innovative Translational Research
  • 2021/12 - 現在 Gifu University United Graduate School of Drug Discovery and Medical Information Sciences
  • 2017/04 - 現在 Gifu University Graduate School of Natural Science and Technology
  • 2008 - 現在 Gifu University Faculty of Engineering
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Awards (3)：
  • 2021/02 - 有機合成化学協会 味の素研究企画賞 カルベンを利用した核酸オリゴマーの実用的合成法の開発
  • 2015/07 - 日本薬学会東海支部 学術奨励賞 核酸医薬開発を目指した化学修飾核酸の創製
  • 2014/08 - 有機合成化学協会東海支部 奨励賞 次世代医薬創出のためのPET標識化法の開発
Association Membership(s) (8)：
The Japanese Biochemical Society ,  The Japan Society of Nucleic Acids Chemistry ,  The Society of Synthetic Organic Chemistry, Japan ,  The Japanese Society for Process Chemistry ,  Japanese Society for Chemical Biology ,  The Chemical Society of Japan ,  American Chemical Society ,  The Pharmaceutical Society of Japan
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