Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABA<sub>B</sub> Receptor Agonist, by the Introduction of a Cyclopropane Ring.

SHUTO S; SHIBUYA N; YAMADA S; OHKURA T; KIMURA R; MATSUDA A

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J-GLOBAL ID：200902155818372596 Reference number：99A0753437

Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABA_B Receptor Agonist, by the Introduction of a Cyclopropane Ring.

強力なGABA_B受容体アゴニストであるバクロフェンのシクロプロパン環の導入により立体配座的に拘束された類似体の合成

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Material：
Volume： 47 Issue： 8 Page： 1188-1192 Publication year： Aug. 15, 1999
JST Material Number： G0504A ISSN： 0009-2363 CODEN： CPBTAL Document type： Article
Article type：短報 Country of issue： Japan (JPN) Language： ENGLISH (EN)

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Aromatic monocyclic carboxylic,peroxycarboxylic,and thiocarboxylic acids , Synthesis of drugs

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Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABAB Receptor Agonist, by the Introduction of a Cyclopropane Ring.

Synthesis of Conformationally Restricted Analogs of Baclofen, a Potent GABA_B Receptor Agonist, by the Introduction of a Cyclopropane Ring.