Art

J-GLOBAL ID：201002252760824374   Reference number：10A0052835

PREPARATION OF NEW NITROGEN-BRIDGED HETEROCYCLES. 68. ONE-POT SYNTHESIS OF 4-SUBSTITUTED 5-ACYLTHIENO[3,2-d]THIAZOLE DERIVATIVES

新しい窒素-橋架け複素環の調製 68 4-置換-5-アシルチエノ[3,2-d]-チアゾール誘導体のワンポット合成

Author (4)： KAKEHI Akikazu (Shinshu Univ., Nagano, JPN) ,  SUGA Hiroyuki (Shinshu Univ., Nagano, JPN) ,  OKUMURA Yukihisa (Shinshu Univ., Nagano, JPN) ,  NISHI Takashi (Shinshu Univ., Nagano, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 81  Issue： 1  Page： 175-184  Publication year： Jan. 01, 2010 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： *nitrogen heterocyclic compound ,  *sulfur heterocyclic compound ,  one-pot synthesis ,  bridged compound ,  reaction mechanism ,  zwitterion ,  by-product ,  Diels-Alder reaction ,  ring-opening reaction ,  cycloaddition ,  ORTEP diagram ,  aromatic carboxylic acid ,  carboxylate (ester) ,  Heterocyclic Compounds, Bridged-Ring ,  Heterocyclic Compounds, 3-Ring ,  Heterocyclic Compounds, 2-Ring ,  retro Diels-Alder reaction ,  *Thiazoles ,  Pyrroles
Semi thesaurus term： *Thiazoles ,  Pyrroles

JST classification (1)： Thiazoles,isothiazoles  (CF07081P)

Substance index (17)： 2-Butynedioic acid dimethyl ,  Phthalic acid dimethyl ,  3-(Pyridinium-1-yl)-4-methyl-5-acetylthiophene-2-thiolate ,  3-(Pyridinium-1-yl)-4-methyl-5-benzoylthiophene-2-thiolate ,  Methyl(6-methylthieno[3,2-d]thiazole-5-yl) ketone ,  Phenyl(6-methylthieno[3,2-d]thiazole-5-yl) ketone ,  4-Chlorophenyl(6-methylthieno[3,2-d]thiazole-5-yl) ketone ,  4-Bromophenyl(6-methylthieno[3,2-d]thiazole-5-yl) ketone ,  Methyl(6-phenylthieno[3,2-d]thiazole-5-yl) ketone ,  Phenyl(6-phenylthieno[3,2-d]thiazole-5-yl) ketone ,  5-(4-Chlorobenzoyl)-6-phenylthieno[3,2-d]thiazole ,  4-Bromophenyl(6-phenylthieno[3,2-d]thiazole-5-yl) ketone ,  2-(5-Acetylthieno[3,2-d]thiazole-6-yl)acetic acid ethyl ester ,  2-(5-Benzoylthieno[3,2-d]thiazole-6-yl)acetic acid ethyl ester ,  2-[5-(4-Chlorobenzoyl)thieno[3,2-d]thiazole-6-yl]acetic acid ethyl ester ,  2-[5-(4-Bromobenzoyl)thieno[3,2-d]thiazole-6-yl]acetic acid ethyl ester ,  2-[(4Z)-7-Acetyl-8-methyl-4H-5,6-dithia-8b-aza-as-indacene-4-ylidene]succinic acid dimethyl ester

Reference (14)：

• For part 67 of this series, see A. Kakehi, H. Suga, Y. Okumura, M. Shinohara, T. Kako, T. Sekiguchi, and M. Shiro, Chem. Pharm. Bull., 2009, 57, 1385.
• L. Grehn, J. Heterocycl. Chem., 1978, 15, 81.
• C. Paulmier, Bull. Soc. Chim. Fr., 1980, 151.
• T. Y. Kvitko, R. V. Khozeeva, N. S. Fedorova, V. A. Sminova, and A. V. El’tsov, Chim. Getro. Soedin., 1979, 474.
• M. Augustin, W. Dölling, and P. Kindt, Zeit. Fuer Chem., 1990, 30, 18.

Terms in the title (7)： 窒素 ,  橋架け ,  複素環 ,  調製 ,  置換 ,  チアゾール誘導体 ,  ワンポット合成