INOKUMA Tsubasa

いのくまつばさ | INOKUMA Tsubasa

Affiliation and department：

Research field (1)： Pharmaceuticals - chemistry and drug development

Research theme for competitive and other funds (9)：

2022 - 2024 Development of the strategy for synthesis of supersulfides based on rationally-designed sulfuration reagent
2022 - 2023 Direct Introduction of Side Chain Structure to Meddle Molecule Peptides and its Application to the Development of Novel Protease Inhibitory Peptides
2020 - 2023 Synthesis of aminophosphoric acid-containing peptides based on direct asymmetric reaction to iminophosphoric acid peptides
2018 - 2020 Asymmetric construction of arylglycine unit and application to the synthesis of unnatural amino acid-containing peptide
2016 - 2018 Novel methodology for the synthesis of unnatural amino acid-containing peptide based on asymmetric construction of indolyl glycine

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Papers (66)：

Tsubasa Inokuma, Ken-ichi Yamada. Improvement of Asymmetric Reactions via Remote Electronic Tuning of N-Heterocyclic Carbene Catalysts. ChemCatChem. 2024. 16. e202401078
Tsubasa Inokuma, Ken-ichi Yamada. Remote Electronic Tuning for High-performance N-Heterocyclic Carbene Catalysis. Journal of Synthetic Organic Chemistry, Japan. 2024. 82. 3. 222-233
Chunzhao Sun, Tsubasa Inokuma, Daisuke Tsuji, Yousuke Yamaoka, Reiko Akagi, Ken-ichi Yamada. Total Synthesis of 1,4a-di-epi-ent-Pancratistatin, Exemplifying a Stereodivergent Approach to Pancratistatin Isomers. Chemical Communications. 2024. 60. 53. 6757-6760
Masayuki Sugano, Tsubasa Inokuma, Yousuke Yamaoka, Ken-ichi Yamada. 5-exo-Selective Asymmetric Bromolactonization of Stilbenecarboxylic Acids Catalyzed by Phenol-bearing Chiral Thiourea. Organic and Biomolecular Chemistry. 2024. 22. 9. 1765-1769
Tsubasa Inokuma, Ken-ichi Yamada. Remote Electronic Tuning of Chiral N-Heterocyclic Carbenes. The Chemical Record. 2023

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MISC (28)：

Daishiroh Kobayashi, Kohdai Nishida, Tsubasa Inokuma, Akira Shigenaga, Akira Otaka. Lossen rearrangement-mediated preparation of N-glyoxylyl peptide without addition of oxidant,. Peptide Science 2019. 2020. 59
Taiki Kohiki, Yusuke Kato, Masaya Denda, Yusuke Nishikawa, Kazuko YORITA, Ikuko Sagawa, Tsubasa Inokuma, Akira Shigenaga, Kiyoshi Fukui, Akira Otaka. Development and application of novel protein labeling reagent "SEAL". Peptide Science 2018. 2019. 104-104
Chiaki Komiya, Jun Tsukimoto, Masahiro Ueda, Takuya Morisaki, Tsubasa Inokuma, Akira Shigenaga, Kouji Itou, Akira Otaka. Preparation of protein thioesters enabled by carboxypeptidase-mediated C-terminal specific hydrazinolysis. Peptide Science 2018. 2019. 8-8
Naoto Naruse, Kento Ohkawachi, Tsubasa Inokuma, Akira Shigenaga, Akira Otaka. N-S-acyl-transfer-mediated On-resin Formation of Thioester with Practical Application to Peptide Synthesis. Peptide Science 2017. 2018. 32-33
Chiaki Komiya, Jun Tsukimoto, Takuya Morisaki, Yusuke Tsuda, Rin Miyajima, Tsubasa Inokuma. Development of methodology for producing thioesters from naturally occurring peptide sequence. Peptide Science 2017. 2018. 86-87

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Lectures and oral presentations (195)：

Development of a synthetic methodology to obtain both epimers of a-indolylglycine-containing peptide in one step
(第61回ペプチド討論会 2024)
硫黄原子の段階的伸長反応による超硫黄分子の新規合成法開発
(第50回反応と合成の進歩シンポジウム 2024)
スチルベンカルボン酸のブロモラクトン化反応における位置選択性制御
(第50回反応と合成の進歩シンポジウム 2024)
含窒素複素環式カルベン触媒を用いるイノシトール合成法を基盤とする立体異性体の網羅的合成を志向した1,4a-di-epi-ent-Pancratistatinの合成
(第53回複素環化学討論会 2024)
含窒素複素環式カルベン触媒を用いる新規チオエステル合成法
(第53回複素環化学討論会 2024)

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Education (3)：

2008 - 京都大学大学院薬学研究科博士後期課程中途退学
2007 - 京都大学大学院薬学研究科修士課程修了
2005 - 京都大学薬学部総合薬学科卒業

Professional career (1)：

博士(薬学) (京都大学)

Work history (7)：

2022/04 - 現在 The University of Tokushima
2017/04 - 2022/03 The University of Tokushima
2015/04 - 2017/03 The University of Tokushima
2013/09 - 2015/03 The University of Tokushima
2012/01 - 2013/08 The Scripps Research Institute

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Committee career (2)：

2021/04 - 2023/03 日本薬学会ファルマシアトピックス小委員
2018/04 - 2020/03 科学技術予測センター専門調査員

Awards (5)：

2021/10 - 徳島県令和3年度徳島県科学技術大賞(若手研究者部門)
2020/12 - 令和2年度徳島大学若手研究者学長表彰多様な側鎖構造をもつ異常アミノ酸類縁体およびペプチド群の効率的かつ迅速合成法の開発
2020/03/25 - The Pharmaceutical Society of Japan 2020年度日本薬学会奨励賞 Synthesis of non-canonical amino acids and peptides containing them for establishment of the template for drug discovery
2017/10/21 - 日本薬学会中国四国支部平成29年度日本薬学会中国四国支部奨励賞ペプチドへの直接的不斉反応を基盤とした非天然アミノ酸含有ペプチドの新規効率的不斉合成法開発
2016/12 - The Society of Synthetic Organic Chemistry,Japan 塩野義製薬研究企画賞ペプチドへの直接的不斉マンニッヒ反応を基盤とする新規効率的中分子合成法の開発

Association Membership(s) (5)：

American Chemical Society , The Japanese Peptide Society , The Society of Synthetic Organic Chemistry,Japan , The Pharmaceutical Society of Japan , 日本ケミカルバイオロジー学会

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