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J-GLOBAL ID：202002226932326128   Reference number：20A0541200

SYNTHESIS AND EVALUATION FOR BIOLOGICAL ACTIVITIES OF 2-THIO-ACYLATED THIAZOLES CONTAINING PYRAZOLE MOIETY

ピラゾール部分を有する2-チオ-アシル化チアゾール類の合成と生物活性の評価

Author (5)： MASUMOTO Eiichi (Fukuoka Univ., Fukuoka, JPN) ,  KASHIGE Nobuhiro (Fukuoka Univ., Fukuoka, JPN) ,  NAGABUCHI Hayate (Fukuoka Univ., Fukuoka, JPN) ,  OKABE-NAKAHARA Fumi (Fukuoka Univ., Fukuoka, JPN) ,  MARUOKA Hiroshi (Fukuoka Univ., Fukuoka, JPN)
Material： Heterocycles  (International Journal for Reviews and Communications in Heterocyclic Chemistry)
Volume： 98  Issue： 12  Page： 1736-1746  Publication year： Dec. 01, 2019 
JST Material Number： S0966A  ISSN： 0385-5414  CODEN： HTCYAM  Document type： Article
Article type： 短報  Country of issue： Japan (JPN)  Language： ENGLISH (EN)

Thesaurus term： chemical synthesis ,...
Semi thesaurus term： DNA Cleavage ,...

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JST classification (2)： Pyrazoles  (CF07082G) ,  Basic research of antibacterial drugs  (GW17020S)

Substance index (10)： Edaravone ,  5-methyl-2-phenyl-4-[2-(thiophene-2-carbonylsulfanyl)-1,3-thiazol-4-yl]pyrazol-3-yl thiophene-2-carboxylate ,  5-methyl-4-[2-(2-methylbenzoylsulfanyl)-1,3-thiazol-4-yl]-2-phenylpyrazol-3-yl 2-methylbenzoate ,  4-(5-hydroxy-3-methyl-1-phenylpyrazol-4-yl)-3H-1,3-thiazole-2-thione ,  4-[2-(4-chlorobenzoylsulfanyl)-1,3-thiazol-4-yl]-5-methyl-2-phenylpyrazol-3-yl 4-chlorobenzoate ,  4-[2-(4-methoxybenzoylsulfanyl)-1,3-thiazol-4-yl]-5-methyl-2-phenylpyrazol-3-yl 4-methoxybenzoate ,  5-methyl-2-phenyl-4-[2-(propanoylsulfanyl)-1,3-thiazol-4-yl]pyrazol-3-yl propanoate ,  Rhodanine ,  4-[2-(benzoylsulfanyl)-1,3-thiazol-4-yl]-5-methyl-2-phenylpyrazol-3-yl benzoate ,  4-[2-(acetylsulfanyl)-1,3-thiazol-4-yl]-5-methyl-2-phenylpyrazol-3-yl acetate

Reference (17)：

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Terms in the title (5)： ピラゾール ,  アシル化 ,  チアゾール類 ,  生物活性 ,  評価