研究キーワード (6件):
Bioinformatics
, Structure-based virtual screening
, MD simulation
, Fragment molecular orbital method
, Molecular modeling
, Cheminformatics
競争的資金等の研究課題 (3件):
2024 - 2028 癌細胞の代謝リプログラミング依存的な糖鎖修飾と癌微小環境応答の解明
2024 - 2027 FMO/ML-Guided Drug Design: Accelerating Novel Inhibitor Development and Drug Discovery
2021 - 2026 Gタンパク質の超硫黄化による新奇シグナル制御とその生理的意義の解明
論文 (55件):
Kamonpan Sanachai, Kowit Hengphasatporn, Supakarn Chamni, Khanit Suwanborirux, Panupong Mahalapbutr, Yasuteru Shigeta, Supaphorn Seetaha, Kiattawee Choowongkomon, Thanyada Rungrotmongkol. Exploring mimosamycin as a Janus kinase 2 inhibitor: A combined computational and experimental investigation. Computational Biology and Chemistry. 2025
Gissi Novientri, Koji Takeda, Lian Duan, Kowit Hengphasatporn, Yasuteru Shigeta, Cheng Xie, Tsuyoshi Mashima, Shun Hirota. Apoprotein Intermolecular Interactions and Heme Insertion for 3D Domain Swapping in Myoglobin. ACS Omega. 2025
Akiyuki Nishimura, Seiryo Ogata, Xiaokang Tang, Kowit Hengphasatporn, Keitaro Umezawa, Makoto Sanbo, Masumi Hirabayashi, Yuri Kato, Yuko Ibuki, Yoshito Kumagai, et al. Polysulfur-based bulking of dynamin-related protein 1 prevents ischemic sulfide catabolism and heart failure in mice. Nature Communications. 2025
Teerapap Panklai, Prapapan Temkitthawon, Nungruthai Suphrom, Corine Girard, Perle Totoson, Kowit Hengphasatporn, Yasuteru Shigeta, Krongkarn Chootip, Kornkanok Ingkaninan. Nymphaea pubescens Willd. extract and its flavonoid constituents vasodilate rat isolated pulmonary artery via NO-sGC-cGMP pathway. Phytomedicine Plus. 2025
Charin Chandit, Kowit Hengphasatporn, Pattraporn Donsuy, Yasuteru Shigeta, Kittikhun Wangkanont. Structure and catalytic activity of a dihydrofolate reductase-like enzyme from Leptospira interrogans. International Journal of Biological Macromolecules. 2025