研究者
J-GLOBAL ID:201401089160331894
更新日: 2024年01月30日 小阪 孝史
コザカ タカシ | Kozaka Takashi
- Hiroshi Wakabayashi, Hiroshi Mori, Tomo Hiromasa, Norihito Akatani, Anri Inaki, Takashi Kozaka, Yoji Kitamura, Kazuma Ogawa, Seigo Kinuya, Junichi Taki. 125I-labeled 2-[4-(2-iodophenyl)piperidino]cyclopentanol (125I-OI5V) imaging visualized augmented sigma-1 receptor expression according to the severity of myocardial ischemia. Journal of Nuclear Cardiology. 2022
- Hiroshi Wakabayashi, Junichi Taki, Hiroshi Mori, Tomo Hiromasa, Norihito Akatani, Anri Inaki, Takashi Kozaka, Kazuhiro Shiba, Kazuma Ogawa, Seigo Kinuya. Visualization of Dynamic Expression of Myocardial Sigma-1 Receptor After Myocardial Ischemia and Reperfusion Using Radioiodine-Labeled 2-[4-(2-iodophenyl)piperidino]cyclopentanol (OI5V) Imaging. Circulation journal : official journal of the Japanese Circulation Society. 2021. 85. 11. 2102-2108
- Taiki Shigeno, Takashi Kozaka, Yoji Kitamura, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. In vitro and in vivo evaluation of [125/123I]-2-[4-(2-iodophenyl)piperidino]cyclopentanol([125/123I]-OI5V) as a potential sigma-1 receptor ligand for SPECT. Annals of nuclear medicine. 2021. 35. 2. 167-175
- Daisuke Miwa, Yoji Kitamura, Takashi Kozaka, Taiki Shigeno, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. (-)-o-[11 C]methyl-trans-decalinvesamicol ((-)-[11 C]OMDV) as a PET ligand for the vesicular acetylcholine transporter. Synapse (New York, N.Y.). 2020. 74. 11. e22176
- Tuyen Thuy Bich Ho, Alessandro Nasti, Akihiro Seki, Takuya Komura, Hiiro Inui, Takashi Kozaka, Yoji Kitamura, Kazuhiro Shiba, Taro Yamashita, Tatsuya Yamashita, et al. Combination of gemcitabine and anti-PD-1 antibody enhances the anticancer effect of M1 macrophages and the Th1 response in a murine model of pancreatic cancer liver metastasis. Journal for immunotherapy of cancer. 2020. 8. 2
- Kazuma Ogawa, Ryohei Masuda, Kenji Mishiro, Mengfei Wang, Takashi Kozaka, Kazuhiro Shiba, Seigo Kinuya, Akira Odani. Syntheses and evaluation of a homologous series of aza-vesamicol as improved radioiodine-labeled probes for sigma-1 receptor imaging. Bioorganic & medicinal chemistry. 2019. 27. 10. 1990-1996
- Ogawa Kazuma, Masuda Ryohei, Mishiro Kenji, Wang Mengfei, Kozaka Takashi, Shiba Kazuhiro, Kinuya Seigo, Odani Akira. Syntheses and evaluation of azavesamicol homologous as radioiodine labeled probes for sigma-1 receptor imaging. JOURNAL OF NUCLEAR MEDICINE. 2019. 60
- Kazuma Ogawa, Ryohei Masuda, Yoshiaki Mizuno, Akira Makino, Takashi Kozaka, Yoji Kitamura, Yasushi Kiyono, Kazuhiro Shiba, Akira Odani. Development of a novel radiobromine-labeled sigma-1 receptor imaging probe. Nuclear medicine and biology. 2018. 61. 28-35
- Kazuma Ogawa, Atsushi Ishizaki, Kenichiro Takai, Yoji Kitamura, Akira Makino, Takashi Kozaka, Yasushi Kiyono, Kazuhiro Shiba, Akira Odani. Evaluation of Ga-DOTA-(D-Asp)n as bone imaging agents: D-aspartic acid peptides as carriers to bone. Scientific reports. 2017. 7. 1. 13971-13971
- Taiki Shigeno, Takashi Kozaka, Yoji Kitamura, Kazuma Ogawa, Kazuhiro Shiba. Characteristics of 2-[ 4-(2-iodophenyl) piperidino] cyclopenntanon (OI5V) as a new siguma-1 receptor imaging agent. JOURNAL OF NUCLEAR MEDICINE. 2017. 58
- Ogawa Kazuma, Mizuno Yoshiaki, Makino Akira, Masuda Ryohei, Kozaka Takashi, Kitamura Yoji, Kiyono Yasushi, Shiba Kazuhiro, Odani Akira. Development of a radiobromine-labeled compound as a sigma receptor ligand for tumor imaging. JOURNAL OF NUCLEAR MEDICINE. 2016. 57
- Yoji Kitamura, Takashi Kozaka, Daisuke Miwa, Izumi Uno, Mohammad Anwar-Ul Azim, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. Synthesis and evaluation of a new vesamicol analog o-[(11)C]methyl-trans-decalinvesamicol as a PET ligand for the vesicular acetylcholine transporter. Annals of nuclear medicine. 2016. 30. 2. 122-9
- Yoji Kitamura, Takashi Kozaka, Daisuke Miwa, Izumi Uno, Mohammad Anwar-ul Azim, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. Synthesis and evaluation of a new vesamicol analog o-[C-11]methyl-trans-decalinvesamicol as a PET ligand for the vesicular acetylcholine transporter. ANNALS OF NUCLEAR MEDICINE. 2016. 30. 2. 122-129
- Izumi Uno, Takashi Kozaka, Daisuke Miwa, Yoji Kitamura, Mohammad Anwar-ul Azim, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. In Vivo Differences between Two Optical Isomers of Radioiodinated o-iodo-trans-decalinvesamicol for Use as a Radioligand for the Vesicular Acetylcholine Transporter. PLOS ONE. 2016. 11. 1
- Izumi Uno, Takashi Kozaka, Daisuke Miwa, Yoji Kitamura, Mohammad Anwar-Ul Azim, Kazuma Ogawa, Junichi Taki, Seigo Kinuya, Kazuhiro Shiba. In Vivo Differences between Two Optical Isomers of Radioiodinated o-iodo-trans-decalinvesamicol for Use as a Radioligand for the Vesicular Acetylcholine Transporter. PloS one. 2016. 11. 1. e0146719
- Kazuma Ogawa, Yoshiaki Mizuno, Kohshin Washiyama, Kazuhiro Shiba, Naruto Takahashi, Takashi Kozaka, Shigeki Watanabe, Atsushi Shinohara, Akira Odani. Preparation and evaluation of an astatine-211-labeled sigma receptor ligand for alpha radionuclide therapy. Nuclear medicine and biology. 2015. 42. 11. 875-9
- 黒宮 里紗, 菅谷 望, 北村 陽二, 三輪 大輔, 小阪 孝史, 小川 数馬, 内匠 透, 柴 和弘. 15q重複モデルマウスにおける脳内ドーパミン神経系の変化. 日本薬学会年会要旨集. 2015. 135年会. 3. 192-192
- Azim Mohammad Anwar-ul, Kozaka Takashi, Uno Izumi, Miwa Daisuke, Kitamura Yoji, Ogawa Kazuma, Makino Akira, Kiyono Yasushi, Shiba Kazuhiro. The potential of o-bromo-trans-decalinvesamicol as a new PET ligand for vesicular acetylcholine transporter imaging. Synapse. 2014. 68. 10. 445-53
- Azim M. A.-u, Kozaka T, Uno I, Miwa D, Kitamura Y, Ogawa K, Makino A, Kiyono Y, Shiba K. The potential of o-bromo-trans-decalinvesamicol as a new PET ligand for vesicular acetylcholine transporter imaging. Synapse. 2014. 68. 10. 445-453
- Syntheses and In-vitro Evaluation of Tetrahydroaminoacridine (THA) Based Analogues as High Affinity Choline Transporter (HAChT) Imaging Probe. Bangladesh J. Nuclear Med. 2014. 17. 2. 97-102
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